Search Results: Kainate

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Kainate receptor
Rabu, 2025-12-24 11:13:18

Kainate receptors, or kainic acid receptors (KARs), are ionotropic receptors that respond to the neurotransmitter glutamate. They were first identified...

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Kainic acid
Rabu, 2026-04-22 10:42:31

Kainic acid, or kainate, is an acid that naturally occurs in some seaweed. Kainic acid is a potent neuroexcitatory amino acid agonist that acts by activating...

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5-Fluorowillardiine
Kamis, 2026-05-28 06:07:33

selective agonist for the AMPA receptor, with only limited effects at the kainate receptor. It is an excitotoxic neurotoxin when used in vivo and so is rarely...

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GRIK5
Rabu, 2025-10-22 02:32:04

Glutamate receptor, ionotropic kainate 5 is a protein that in humans is encoded by the GRIK5 gene. This gene encodes a protein that belongs to the glutamate-gated...

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Glutamate (neurotransmitter)
Minggu, 2026-05-24 14:36:01

receptors, and metabotropic glutamate receptors. A fourth class, known as kainate receptors, are similar in many respects to AMPA receptors, but much less...

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GYKI 52466
Rabu, 2025-12-24 11:46:49

receptor antagonist (IC50 values are 10-20, ~ 450 and >> 50 μM for AMPA-, kainate- and NMDA-induced responses respectively), orally-active anticonvulsant...

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GRIK2
Selasa, 2026-02-24 06:02:47

Glutamate ionotropic receptor kainate type subunit 2, also known as ionotropic glutamate receptor 6 or GluR6, is a protein that in humans is encoded by...

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Willardiine
Sabtu, 2026-04-04 03:50:57

receptors: AMPA and kainate receptors. Willardiine analogs have been developed that have different binding affinities for the AMPA and kainate receptors. These...

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Tezampanel
Rabu, 2025-12-24 09:39:37

of the AMPA and kainate subtypes of the ionotropic glutamate receptor family, with selectivity for the GluR5 subtype of the kainate receptor. It has...

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SYM-2081
Sabtu, 2025-07-19 02:21:07

selective agonist for the kainate receptor. This potent agonist has nearly 3,000 fold- and 200-fold selectivity for kainate receptors over AMPA and NMDA...

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Ionotropic glutamate receptor
Sabtu, 2026-04-11 21:51:59

binding properties (pharmacology) and sequence similarity: AMPA receptors, kainate receptors, NMDA receptors and delta receptors (see below). AMPA receptors...

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GRIK1
Senin, 2026-01-05 14:04:50

Glutamate receptor, ionotropic, kainate 1, also known as GRIK1, is a protein that in humans is encoded by the GRIK1 gene. This gene encodes one of the...

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AP5
Kamis, 2025-10-16 01:36:37

isolate the action of other glutamate receptors in the brain, i.e., AMPA and kainate receptors. AP5 can block the conversion of a silent synapse to an active...

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5-Iodowillardiine
Sabtu, 2026-05-30 18:49:47

a selective agonist for some kainate receptor subunits with only limited effects at AMPA receptors. It activates kainate receptors containing GluK1 (GluR5)...

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Riluzole
Selasa, 2026-05-26 06:39:37

damaged neurons. Riluzole has also been reported to directly inhibit the kainate and NMDA receptors. The drug has also been shown to postsynaptically potentiate...

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NBQX
Selasa, 2025-12-23 14:03:47

AMPA receptors in micromolar concentrations (~10–20 μM) and also blocks kainate receptors. In experiments, it is used to counter glutamate excitotoxicity...

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N-Methyl-D-aspartic acid
Kamis, 2025-12-11 05:00:07

has no effect on other glutamate receptors (such as those for AMPA and kainate). NMDA receptors are particularly important when they become overactive...

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Quisqualic acid
Jumat, 2026-02-06 12:55:00

Quisqualic acid is an agonist of the AMPA, kainate, and group I metabotropic glutamate receptors. It is one of the most potent AMPA receptor agonists...

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NS102
Kamis, 2024-09-26 21:07:26

NS102 is a kainate receptor antagonist. NS102 at Sigma-Aldrich Johansen, Tina H; Drejer, Joergen; Watjen, Frank; Nielsen, Elsebet O (1993). "A novel non-NMDA...

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Ibotenic acid
Rabu, 2026-05-20 13:40:50

and II metabotropic glutamate receptors, and weakly activating AMPA and kainate receptors. Taken systemically, it is a prodrug of muscimol, broken down...

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Nephila polyamine toxin 8
Senin, 2026-04-13 19:24:27

especially potent at kainate receptors and AMPA receptors, with inhibitory potencies summarised in the table: The inhibition of kainate receptors by NPTX-8...

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GRIK4
Kamis, 2025-07-17 00:27:42

GRIK4 (glutamate receptor, ionotropic, kainate 4) is a kainate receptor subtype belonging to the family of ligand-gated ion channels which is encoded...

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CNQX
Selasa, 2025-12-23 14:04:19

cyanquixaline (6-cyano-7-nitroquinoxaline-2,3-dione) is a competitive AMPA/kainate receptor antagonist. Its chemical formula is C9H4N4O4. CNQX is often used...

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Juan Lerma Gómez
Selasa, 2026-03-10 08:48:18

its role in health and disease. He described the existence of functional kainate receptors (KARs) in central neurons and applied single-cell RT-PCR to study...

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Enflurane
Sabtu, 2026-03-28 19:09:21

and 5-HT3 receptors, and as a negative allosteric modulator of the AMPA, kainate, and NMDA receptors, as well as of nicotinic acetylcholine receptors. Clinically...

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Saffron
Rabu, 2026-05-27 21:56:16

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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NMDA receptor
Kamis, 2026-01-29 23:47:46

types of ionotropic glutamate receptors, the other two being AMPA and kainate receptors. Depending on its subunit composition, its ligands are glutamate...

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Evans blue (dye)
Selasa, 2025-12-23 14:28:44

pharmacologically active, acting as a negative allosteric modulator of the AMPA and kainate receptors and as an inhibitor of vesicular glutamate transporters. It also...

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Theanine
Sabtu, 2026-05-23 21:27:32

ionotropic glutamate receptors in the micromolar range, including the AMPA and kainate receptors and, to a lesser extent, the NMDA receptor. It acts as an antagonist...

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Pregnenolone sulfate
Selasa, 2026-04-07 07:34:24

lesser extent, it also acts as a negative allosteric modulator of the AMPA, kainate, and glycine receptors, and may interact with the nACh receptors as well...

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Neuron
Sabtu, 2026-05-30 00:03:48

is a G-protein coupled receptor (often referred to as GPCR). AMPA and Kainate receptors function as cation channels permeable to Na+ cation channels...

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Dextromethorphan
Kamis, 2026-04-02 19:40:24

et al. (April 2005). "The dextromethorphan analog dimemorfan attenuates kainate-induced seizures via sigma1 receptor activation: comparison with the effects...

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Glutamate receptor
Rabu, 2026-05-20 22:20:23

plasticity. They are activated by the drug kainate and are permeable to both sodium and potassium ions. Kainate receptors are expressed in a variety of brain...

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SN 35210
Sabtu, 2025-12-27 09:00:03

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Kynurenic acid
Rabu, 2026-03-04 00:39:59

to act on five targets: As an antagonist at ionotropic AMPA, NMDA and Kainate glutamate receptors in the concentration range of 0.1-2.5 mM. As a noncompetitive...

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A-NK
Sabtu, 2025-12-27 08:32:51

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Phenobarbital
Sabtu, 2026-05-02 23:36:24

post-synaptic neuron will be increased. Direct blockade of glutamatergic AMPA and kainate receptors are also believed to contribute to the hypnotic/anticonvulsant...

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Diazoxide
Minggu, 2026-05-31 11:04:06

hyperinsulinism. Diazoxide acts as a positive allosteric modulator of the AMPA and kainate receptors, suggesting potential application as a cognitive enhancer. Diazoxide...

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Reversal potential
Sabtu, 2025-12-20 20:44:18

neurotransmitter receptors including glutamate receptors (AMPA, NMDA, and kainate), nicotinic acetylcholine (nACh), and serotonin (5-HT3) receptors are nonselective...

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Β-Methylamino-L-alanine
Senin, 2026-03-09 11:24:09

excitotoxin on glutamate receptors, such as NMDA, calcium-dependent AMPA, and kainate receptors. The activation of the metabotropic glutamate receptor 5 is believed...

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Proline
Kamis, 2026-05-07 03:55:27

weak agonist of the glycine receptor and of both NMDA and non-NMDA (AMPA/kainate) ionotropic glutamate receptors. It has been proposed to be a potential...

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GRIK3
Selasa, 2025-07-15 11:13:27

Glutamate receptor, ionotropic kainate 3 is a protein that in humans is encoded by the GRIK3 gene. This gene encodes a protein that belongs to the ligand-gated...

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Quisqualamine
Minggu, 2025-12-21 17:15:08

vitro. The NMDA receptor antagonists magnesium and DL-AP5, the AMPA and kainate receptor antagonist CNQX, and the GABAB receptor antagonist 2-hydroxysaclofen...

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Barbiturate
Selasa, 2026-04-28 05:16:03

In addition to this GABAergic effect, barbiturates also block AMPA and kainate receptors, subtypes of ionotropic glutamate receptor. Glutamate is the...

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Furosemide
Jumat, 2026-05-22 17:55:16

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Hexobarbital
Jumat, 2025-03-21 22:45:52

inhibitory effect, hexobarbital blocks, like all barbiturates, AMPA receptors, kainate receptors, neural acetylcholine receptors. And above all, barbiturates...

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AMPA receptor
Rabu, 2026-05-06 12:02:46

"Structure of a glutamate-receptor ligand-binding core in complex with kainate". Nature. 395 (6705): 913–7. Bibcode:1998Natur.395..913A. doi:10.1038/27692...

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F-17475
Sabtu, 2026-02-21 12:50:13

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Phenidone
Minggu, 2026-05-03 23:26:53

Myung-Bok; Kim, Won-Ki; Ko, Kwang Ho (August 18, 2000). "Phenidone prevents kainate-induced neurotoxicity via antioxidant mechanisms". Brain Research. 874...

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Atomoxetine
Selasa, 2026-06-02 14:48:14

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Glutamine
Sabtu, 2026-01-10 19:31:32

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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UBP-302
Jumat, 2026-01-02 00:04:02

UBP-302 is a highly selective kainate receptor antagonist used in the study of many neurological processes. It is active at micromolar concentration within...

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Serotonin
Jumat, 2026-06-05 15:37:48

neurons increase with intense visual stimuli. Animal models suggest that kainate signaling negatively regulates serotonin actions in the retina, with possible...

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Nitrous oxide
Kamis, 2026-05-07 21:34:49

blocks NMDAR and β2-subunit-containing nACh channels, weakly inhibits AMPA, kainate, GABAC and 5-HT3 receptors, and slightly potentiates GABAA and glycine...

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Glossary of neuroscience
Rabu, 2026-01-21 21:24:09

processing during sleep. Kainate receptor A subtype of ionotropic glutamate receptor involved in fast excitatory synaptic transmission. Kainate receptors play roles...

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List of investigational headache and migraine drugs
Jumat, 2026-06-05 11:36:24

– migraine [77] Dasolampanel (NGX-426) – ionotropic glutamate AMPA and kainate receptor antagonist – migraine [78] Dextromethorphan/quinidine (DXM/Q;...

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Trifluoromethyldeschloroketamine
Sabtu, 2025-12-27 09:01:33

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Methadone
Selasa, 2026-06-02 22:13:18

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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2F-NENDCK
Senin, 2026-05-04 19:38:35

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Spermidine
Selasa, 2026-02-17 23:56:19

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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SePP
Senin, 2026-02-23 11:15:53

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ibogaine
Minggu, 2026-06-07 05:07:29

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Chloroform
Senin, 2026-04-13 03:17:56

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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3-Me-PCE
Kamis, 2026-02-12 03:56:47

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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SGK1
Selasa, 2026-02-24 06:07:42

role of SGK1 in memory consolidation. "SGK isoforms upregulate AMPA and kainate receptors and thus are expected to enhance the excitatory effects of glutamate"...

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Diphenidine
Sabtu, 2026-02-14 15:30:54

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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NMDA receptor antagonist
Kamis, 2026-04-02 22:11:23

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Amantadine
Rabu, 2026-01-07 06:44:28

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Food noise
Rabu, 2026-05-27 04:14:54

receptor signaling in the ventral tegmental area are mediated by AMPA/kainate receptors". American Journal of Physiology. Endocrinology and Metabolism...

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MDPCP
Minggu, 2026-05-17 22:18:27

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Sodium thiopental
Rabu, 2026-02-25 02:52:02

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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G protein-coupled receptor
Senin, 2026-06-01 17:51:25

receptor, 5-HT3 serotonin receptor and glutamate receptors (NMDAR, AMPAR and kainate receptor), which are ion channels. Regulation of immune system activity...

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Dehydroepiandrosterone
Jumat, 2026-01-30 21:53:59

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Dextropropoxyphene
Selasa, 2026-06-02 14:48:46

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Aspartic acid
Kamis, 2026-03-26 02:34:58

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Domoic acid
Rabu, 2026-04-22 10:43:25

and amygdaloid nucleus. It damages the neurons by activating AMPA and kainate receptors, causing an influx of calcium. Although calcium flowing into...

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Calsequestrin
Sabtu, 2025-05-24 05:36:54

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Halothane
Selasa, 2026-01-27 04:51:36

activates 5-HT3 and twin-pore K+ channels. It does not affect the AMPA or kainate receptors. Halothane (2-bromo-2-chloro-1,1,1-trifluoroethane) is a very...

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Methylene blue
Jumat, 2026-05-22 06:54:00

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Glutamic acid
Rabu, 2026-06-03 16:35:07

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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List of investigational tinnitus drugs
Kamis, 2026-05-14 06:57:15

[13] Selurampanel (BGG-492; BGG-492A) – ionotropic glutamate AMPA and kainate receptor antagonist [14] Sodium phenylbutyrate slow-release (4-PB-D-alanin;...

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Lacosamide
Selasa, 2026-05-19 21:16:52

abnormal neuronal connections in the brain. Lacosamide does not affect AMPA, kainate, NMDA, GABAA, GABAB or a variety of dopaminergic, serotonergic, adrenergic...

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Neurotransmitter
Kamis, 2026-05-28 23:46:44

acids Glutamate Glu, E Metabotropic glutamate receptors NMDA receptors, kainate receptors, AMPARs Small: Amino acids Gamma-aminobutyric acid GABA GABAB...

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Pethidine
Sabtu, 2026-05-23 07:49:18

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ketamine
Jumat, 2026-05-08 01:06:57

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Chain reactions in living organisms
Selasa, 2025-10-14 23:26:55

during seizure — Evidence from 13C-enrichment of extracellular glutamate in kainate rat model". PLOS ONE. 12 (4) e0174845. Bibcode:2017PLoSO..1274845K. doi:10...

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Neurotransmitter receptor
Kamis, 2026-05-07 13:18:50

GABAA, GABAB1a, GABAB1δ, GABAB2, GABAA-rho Glutamatergic: NMDA, AMPA, Kainate, mGluR1, mGluR2, mGluR3, mGluR4, mGluR5, mGluR6, mGluR7 Glycinergic: Glycine...

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Sevoflurane
Rabu, 2026-05-06 00:38:18

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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NMDA receptor modulator
Minggu, 2026-02-08 03:05:21

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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2-Fluorodeschloroketamine
Minggu, 2026-03-15 13:51:43

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Topiramate
Rabu, 2026-05-27 04:46:05

channels, high-voltage-activated calcium channels, GABAA receptors, AMPA/kainate receptors, and carbonic anhydrase isoenzymes. There is evidence that topiramate...

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Nitrous oxide (medication)
Sabtu, 2026-02-14 03:50:17

blocks NMDAR and β2-subunit-containing nACh channels, weakly inhibits AMPA, kainate, GABAC and 5-HT3 receptors, and slightly potentiates GABAA and glycine...

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Teresa Puthussery
Minggu, 2026-04-26 08:34:20

Venkataramani, S., Gayet-Primo, J., Grünert, U., & Taylor, W. R. (2014). Kainate Receptors Mediate Synaptic Input to Transient and Sustained OFF Visual...

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BQ-869
Rabu, 2026-04-22 14:42:05

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Tiletamine
Senin, 2026-03-16 00:30:08

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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FBLN5
Sabtu, 2025-07-19 12:48:06

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Retigabine
Minggu, 2026-05-31 10:59:29

electroshock, electrical kindling of the amygdala, pentylenetetrazol, kainate, NMDA, and picrotoxin. Researchers hoped this wide-ranging activity would...

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3-Fluorodeschloroketamine
Sabtu, 2025-12-27 08:21:51

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Astrocyte
Selasa, 2026-05-19 10:08:25

(α-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid), NMDA (N-methyl-D-aspartate) and kainate subtypes of ionotropic glutamate receptors follows. It is the activation...

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Hydrochlorothiazide
Rabu, 2026-05-13 18:25:57

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Glutathione
Senin, 2026-05-11 06:30:11

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Diethyl ether
Selasa, 2026-06-02 15:32:44

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Cyclothiazide
Rabu, 2025-12-24 09:55:44

that cyclothiazide is a positive allosteric modulator of the AMPA and kainate receptors, capable of reducing or essentially eliminating rapid desensitization...

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CNS-5161
Senin, 2026-02-09 11:46:37

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ketamir-2
Sabtu, 2026-02-21 12:27:28

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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NETO1
Kamis, 2025-12-18 19:07:59

positive regulation of excitatory postsynaptic potential regulation of kainate selective glutamate receptor activity Sources:Amigo / QuickGO Orthologs...

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Selurampanel
Jumat, 2026-01-30 10:03:52

quinoxalinedione series which acts as a competitive antagonist of the AMPA and kainate receptors and, as of 2015, is being investigated in clinical trials by...

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Osavampator
Minggu, 2026-03-22 15:00:46

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Gunnar Svaetichin
Rabu, 2025-10-01 04:51:33

(March 1984). "Hyperpolarization of fish retinal horizontal cells by kainate and quisqualate". Nature. 308 (5957): 360–362. Bibcode:1984Natur.308..360H...

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Acromelic acid A
Kamis, 2025-07-17 22:08:38

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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2-Oxo-PCE
Senin, 2026-05-04 19:38:33

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Memantine
Kamis, 2026-05-28 07:16:07

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Fluorexetamine
Sabtu, 2025-12-27 08:20:30

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Xenon
Selasa, 2026-06-02 01:14:34

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Calcium signaling
Kamis, 2026-06-04 02:04:03

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Acetylcysteine
Kamis, 2026-04-02 02:17:58

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Radu Aricescu
Rabu, 2025-10-01 12:01:01

complexes", Science, vol. 353, issue 6296 (2016). "Transsynaptic Modulation of Kainate Receptor Functions by C1q-like Proteins", Neuron, vol. 90, issue 4 (2016)...

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Meprobamate
Rabu, 2026-02-04 14:24:32

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Carisoprodol
Selasa, 2026-05-05 06:04:28

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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3-Methyl-PCP
Sabtu, 2025-12-27 08:31:39

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Zinc
Jumat, 2026-06-05 21:56:22

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Syntenin-1
Jumat, 2025-07-18 01:31:12

Couthino V (February 2003). "Rapid and differential regulation of AMPA and kainate receptors at hippocampal mossy fibre synapses by PICK1 and GRIP". Neuron...

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Neurocalcin
Jumat, 2026-02-20 06:15:35

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Piracetam
Kamis, 2026-03-26 03:39:30

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Hemantane
Sabtu, 2026-03-14 19:21:08

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Allopregnanolone
Selasa, 2026-05-12 05:45:06

no action at other ligand-gated ion channels, including the NMDA, AMPA, kainate, and glycine receptors. Unlike progesterone, allopregnanolone is inactive...

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Xanthurenic acid
Selasa, 2025-12-23 12:02:44

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Dimemorfan
Kamis, 2025-05-29 21:18:05

et al. (April 2005). "The dextromethorphan analog dimemorfan attenuates kainate-induced seizures via sigma1 receptor activation: comparison with the effects...

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2-Bromodeschloroketamine
Sabtu, 2025-12-27 08:34:01

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Esketamine
Sabtu, 2026-05-02 02:22:03

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Convulsant
Rabu, 2026-02-04 13:01:58

in animals as it is a cyclic analog of l-glutamate and an agonist for kainate receptors in the brain which makes it a potent neurotoxin and excitant...

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NEFA (drug)
Sabtu, 2025-12-27 07:09:49

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Haloperidol
Selasa, 2026-06-02 14:49:07

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Dizocilpine
Senin, 2026-04-27 11:28:08

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Alexei Verkhratsky
Senin, 2026-03-02 11:40:51

Kettenmann, H.; Verkhratsky, A. (1997). "Na+/Ca2+ exchanger modulates kainate-triggered Ca2+ signaling in Bergmann glial cells in situ". FASEB J. 11...

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Amnesic shellfish poisoning
Sabtu, 2024-09-14 16:11:48

and amygdaloid nucleus. It damages the neurons by activating AMPA and kainate receptors, causing an influx of calcium. Although calcium flowing into...

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Magnesium
Kamis, 2026-05-28 20:39:07

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Eliprodil
Senin, 2026-05-11 13:59:45

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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DLG4
Kamis, 2025-07-31 20:47:58

Couthino V (February 2003). "Rapid and differential regulation of AMPA and kainate receptors at hippocampal mossy fibre synapses by PICK1 and GRIP". Neuron...

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EVT-103
Jumat, 2024-01-05 14:19:53

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Deoxymethoxetamine
Sabtu, 2025-12-27 08:35:25

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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GRIA2
Senin, 2025-10-27 23:17:06

specifically the ionotropic AMPA receptor subunits (GluR2, GluR3, GluR4) and kainate receptor subunits (GluR5, GluR6). Glutamate-gated ion channels are composed...

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Nitric oxide
Selasa, 2026-05-26 13:14:18

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Biological neuron model
Selasa, 2026-05-12 12:06:45

kinetic currents. Four neurotransmitters primarily influence the CNS. AMPA/kainate receptors are fast excitatory mediators while NMDA receptors mediate considerably...

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Annexin
Kamis, 2026-01-01 08:54:05

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Dextromethorphan/bupropion
Kamis, 2026-06-04 15:43:12

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Alcohol (drug)
Senin, 2026-06-01 02:31:31

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Glycine
Senin, 2026-04-27 18:18:56

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Dimethylglycine
Senin, 2026-05-04 00:02:11

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Alanine
Kamis, 2026-04-30 13:17:28

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Phencyclidine
Jumat, 2026-05-15 14:16:34

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Philanthotoxin
Jumat, 2026-01-30 09:58:45

Philanthotoxins reversibly inhibit AMPA (also called the "quisqualate receptor"), kainate, and NMDA ionotropic glutamate receptors (iGluRs). Philanthotoxins have...

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Blixeprodil
Senin, 2026-05-04 19:48:10

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Toluene
Jumat, 2026-04-24 10:24:19

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Dasolampanel
Selasa, 2025-12-23 14:23:19

analog of tezampanel and thereby competitive antagonist of the AMPA and kainate receptors which was under development by Raptor Pharmaceuticals/Torrey...

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Putrescine
Senin, 2026-01-26 14:51:19

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Edward Boyden
Selasa, 2026-05-19 06:02:11

high-efficacy soma-targeted opsin through combining the N-terminal 150 residues of kainate receptor subunit 2 (KA2) to the high-photocurrent channelrhodopsin CoChR...

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L-701324
Sabtu, 2025-12-27 19:02:22

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Theanne Griffith
Sabtu, 2025-12-27 01:11:16

Swanson G (2015). "Identification of critical functional determinants of kainate receptor modulation by auxiliary protein Neto2". Journal of Physiology...

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Tramadol
Jumat, 2026-05-29 05:45:43

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Farampator
Kamis, 2026-06-04 09:25:58

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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S-phase kinase-associated protein 1
Sabtu, 2025-07-19 14:21:56

SCF-like ubiquitin ligase complex and protects postmitotic neurons from kainate excitotoxicity". Neuron. 37 (5): 735–49. doi:10.1016/s0896-6273(03)00084-9...

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3-Methyl-PCPy
Sabtu, 2025-12-27 08:51:12

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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GRID2
Minggu, 2025-12-28 20:07:35

glutamate receptors. They possess 14–24% sequence homology with AMPA, kainate, and NMDA subunits, but, despite their name, have been found not to directly...

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CX1739
Senin, 2026-03-30 14:10:56

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Chromosome 21
Minggu, 2025-09-28 04:19:32

protein 3A, mitochondrial GRIK1: encoding glutamate receptor ionotropic, kainate 1 H2BC12L: encoding histone H2B type F-S HLCS: encoding enzyme holocarboxylase...

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Northern blot
Jumat, 2026-01-02 02:42:24

Zukin, R. S. (1993). "Developmental Regulation of mRNAs Encoding Rat Brain Kainate/AMPA Receptors: A Northern Analysis Study". J. Neurochem. 61 (6): 2239–2246...

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L-687,414
Sabtu, 2026-02-21 15:01:44

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Long-term depression
Sabtu, 2026-05-30 04:20:50

α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid receptors (AMPARs), kainate receptors (KARs), and metabotropic glutamate receptors (mGluRs) during...

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Mibampator
Selasa, 2025-12-23 11:54:57

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Diethylenetriamine
Jumat, 2026-06-05 14:21:21

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Inhalational anesthetic
Rabu, 2026-05-13 06:02:09

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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AMPA receptor positive allosteric modulator
Selasa, 2025-12-23 11:54:16

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Pentobarbital
Rabu, 2026-05-20 22:50:26

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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DNQX
Selasa, 2025-12-23 14:04:07

7-dinitroquinoxaline-2,3-dione) is a competitive antagonist at AMPA and kainate receptors, two ionotropic glutamate receptor (iGluR) subfamilies. It is...

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Channel blocker
Rabu, 2025-12-24 13:02:13

Channel blockers are also known to act at AMPA receptors, Glycine receptors, Kainate receptors, P2X receptors and Zinc (Zn2+)-activated channels. The type of...

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ACEA-1328
Rabu, 2025-12-24 23:52:43

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Hydroxetamine
Sabtu, 2025-12-27 08:47:28

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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1-Aminocyclopropane-1-carboxylic acid
Senin, 2025-11-24 05:28:30

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Pharmacology of ethanol
Minggu, 2026-04-05 14:07:08

negative allosteric modulator AMPA receptor: negative allosteric modulator Kainate receptor: negative allosteric modulator Glycine receptor: positive allosteric...

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Lanicemine
Rabu, 2025-12-24 11:08:21

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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3-Chloro-PCP
Minggu, 2026-05-17 02:28:14

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Kynurenine
Kamis, 2026-03-12 04:56:20

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Farah Lubin
Minggu, 2026-04-12 18:59:26

expression and transcriptional regulation in the hippocampus. She found that kainate, a glutamate analog, elicited activation of NF-κB via the classical IkB...

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Spermine
Sabtu, 2026-02-21 22:41:33

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ketamine/temsirolimus
Jumat, 2025-02-28 12:11:07

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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AMPA
Selasa, 2025-02-11 02:25:59

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Trichloroethylene
Kamis, 2026-06-04 09:43:04

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Deschloroketamine
Sabtu, 2025-12-27 08:34:36

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Radiprodil
Senin, 2026-01-26 14:02:36

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Minocycline
Kamis, 2026-06-04 16:40:01

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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NYX-2925
Senin, 2026-02-23 11:52:45

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Excitatory synapse
Kamis, 2025-09-18 06:51:07

postsynaptic receptors including the NMDA receptor, AMPA receptor, and kainate receptors. These receptors are all cation channels that allow positively...

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3-Fluoro-PCP
Senin, 2026-05-04 19:38:37

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Bumetanide
Selasa, 2026-03-03 01:57:01

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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GRIA3
Senin, 2025-10-27 23:16:02

ionotropic AMPA glutamate receptor subunits (GluA2, GluA3, GluA4) and kainate receptor subunits (GluK1, GluK2). Glutamate gated ion channels are made...

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Receptor (biochemistry)
Sabtu, 2026-05-16 00:35:41

Receptors G protein Exogenous Ligand Glutamate iGluRs: NMDA, AMPA, and Kainate receptors Na+, K+, Ca2+ Ketamine Glutamate receptors: mGluRs Gq or Gi/o...

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Cytidine
Selasa, 2026-04-07 12:17:09

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Silent synapse
Senin, 2026-03-30 07:56:17

(AMPARs) (formerly known as quisqualate receptors), NMDA receptors (NMDARs), kainate receptors, and metabotropic glutamate receptors (mGluRs). Most research...

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S100 protein
Sabtu, 2025-10-04 15:18:15

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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NPDPA
Sabtu, 2026-02-21 18:47:24

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Orphenadrine
Selasa, 2026-06-02 14:49:37

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Excitatory amino acid receptor ligand
Jumat, 2024-03-22 12:39:12

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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HA-966
Minggu, 2025-12-21 15:58:19

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Nooglutyl
Kamis, 2026-06-04 01:03:58

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Cyclic glycine-proline
Minggu, 2025-12-21 13:13:58

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Methoxyflurane
Sabtu, 2026-02-21 17:05:10

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Methoxpropamine
Kamis, 2026-01-01 17:31:19

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Annexin A1
Senin, 2025-11-17 11:25:01

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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18-Methoxycoronaridine
Senin, 2026-05-11 19:16:26

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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1,1,1-Trichloroethane
Jumat, 2026-02-27 20:03:58

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Oligodendrocyte progenitor cell
Sabtu, 2025-10-04 23:28:52

proteoglycan-positive oligodendrocyte precursor cells in the normal and kainate-lesioned rat hippocampus". Neuroscience. 92 (1): 83–95. doi:10.1016/S0306-4522(98)00751-9...

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Ketofol
Rabu, 2025-05-28 23:27:11

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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2-FXPr
Sabtu, 2025-12-27 08:26:31

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Huperzine A
Minggu, 2026-05-17 02:28:01

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Halogenated ether
Jumat, 2026-05-15 22:56:07

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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FBXW7
Kamis, 2025-07-17 23:34:08

SCF-like ubiquitin ligase complex and protects postmitotic neurons from kainate excitotoxicity". Neuron. 37 (5): 735–49. doi:10.1016/s0896-6273(03)00084-9...

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Ligand-gated ion channel
Senin, 2025-10-27 23:27:58

HBGR2 GLUA3, GluR3, GluRC, GluR-C, GluR-K3 GLUA4, GluR4, GluRD, GluR-D Kainate GluK GluK1 GluK2 GluK3 GluK4 GluK5 GRIK1 GRIK2 GRIK3 GRIK4 GRIK5 GLUK5...

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List of investigational substance-related disorder drugs
Jumat, 2026-06-05 08:37:19

Tezampanel (LY-293558; NGX-424; PRN-001-01) – ionotropic glutamate AMPA and kainate receptor antagonist – opioid-related disorders TMP-301 (Heptares 25; HTL-0014242;...

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Apigenin
Kamis, 2026-06-04 14:44:26

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Biology of bipolar disorder
Senin, 2026-05-25 04:45:44

and neuronal morphology. The rACC demonstrates reduced expression NMDA, kainate and GABA related proteins. These findings may be compensating for increased...

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Pramiracetam
Jumat, 2025-11-21 09:38:48

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Psychotridine
Rabu, 2025-12-24 12:05:45

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Membrane estrogen receptor
Kamis, 2026-05-21 15:53:46

(February 1998). "Novel mechanism for non-genomic action of 17β-oestradiol on kainate-induced currents in isolated rat CA1 hippocampal neurones". The Journal...

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Quinoxalinedione
Selasa, 2025-12-23 14:02:36

for the diol tautomer. Quinoxalinediones act as antagonists of the AMPA, kainate, and/or NMDA receptors of the ionotropic glutamate receptor family. Examples...

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Calbindin
Selasa, 2025-12-30 20:39:40

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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David Lodge (scientist)
Sabtu, 2024-10-19 19:40:04

characterised its actions between AMPA, N-Methyl-D-aspartic acid (NMDA) and kainate receptor subtypes. At the Royal Veterinary College, Lodge linked his interests...

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Agmatine
Senin, 2026-03-23 06:45:50

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Dextrorphan
Minggu, 2026-04-26 20:47:44

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Tyrosine phosphorylation
Sabtu, 2025-06-14 12:30:34

receptors. These receptors can be divided into three major classes, AMPA, kainate, and NMDA receptors, based on their selective agonists and on their physiological...

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Inositol trisphosphate
Senin, 2025-10-13 09:58:47

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Molecular neuroscience
Selasa, 2024-04-02 02:05:51

concentrations. Ionotropic glutamate receptors can include NMDA, AMPA, and kainate receptors. These receptors are named after agonists that facilitate glutamate...

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Lomerizine
Jumat, 2026-01-23 16:41:24

protection against NMDA-induced and kainate-induced neurotoxicity. Lomerizine was shown to have little affinity for NMDA or kainate receptors, so its protectivity...

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Bita Moghaddam
Rabu, 2026-05-13 23:32:16

local activation of ionotropic glutamate receptors (AMPA receptors and kainate receptors). A few years later, she found that metabotropic glutamate receptors...

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Changjoon Justin Lee
Selasa, 2025-12-23 09:01:11

Reese Hospital, Columbia University Thesis The Expression and Function of Kainate and AMPA Receptors in Nociceptive Dorsal Root Ganglion Neurons  (2001)...

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Clavulanic acid
Sabtu, 2026-05-30 18:29:58

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Indeloxazine
Rabu, 2026-05-27 04:23:00

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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1,2-Diphenylethylamine
Sabtu, 2026-02-21 12:57:20

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Aniracetam
Minggu, 2025-03-30 22:17:03

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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ZD-9379
Senin, 2025-12-29 22:03:09

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Apimostinel
Senin, 2025-06-30 21:43:30

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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CGP-39551
Sabtu, 2025-12-27 02:50:18

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ana Cristina Rego
Sabtu, 2026-06-06 02:02:43

(11-12), 1405-1417 AC Rego, MW Ward, DG Nicholls. Mitochondria control ampa/kainate receptor-induced cytoplasmic calcium deregulation in rat cerebellar granule...

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Dextromethorphan/quinidine
Senin, 2025-12-15 15:00:15

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Gliotransmitter
Senin, 2025-09-08 21:12:03

cytosolic Ca2+ concentrations in astrocytes. Its main target receptors include Kainate receptors, metabotropic glutamate receptors (mGluRs), and especially N-methyl...

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Microglia
Rabu, 2026-05-20 14:41:29

Christensen RN, Ha BK, Sun F, Bresnahan JC, Beattie MS (July 2006). "Kainate induces rapid redistribution of the actin cytoskeleton in ameboid microglia"...

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Osteocalcin
Rabu, 2026-04-22 21:36:11

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Cycloserine
Rabu, 2026-05-27 15:25:19

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Stephen Heinemann
Jumat, 2025-07-18 01:28:11

Heinemann contributed to differentiating: AMPA receptors, NMDA receptors, and kainate receptors. As shown by Heinemann, NMDA receptors differ in that they allow...

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Perampanel
Kamis, 2026-05-14 14:50:07

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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PCPEP
Sabtu, 2025-12-27 08:56:13

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ampakine
Rabu, 2025-12-24 08:38:37

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Pre-Bötzinger complex
Selasa, 2026-04-07 06:23:58

studies showed that excitatory transmission, predominantly via AMPA- and kainate-type ionotropic glutamate receptors were essential for rhythm generation...

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Delucemine
Sabtu, 2025-12-27 07:10:55

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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GRIA1
Senin, 2025-10-27 23:16:29

2003). "Heteromer formation of delta2 glutamate receptors with AMPA or kainate receptors". Brain Res. Mol. Brain Res. 110 (1): 27–37. doi:10.1016/s0169-328x(02)00561-2...

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4-Keto-PCP
Sabtu, 2025-12-27 08:32:11

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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DLG3
Kamis, 2025-07-17 23:21:41

Garcia EP, Mehta S, Blair LA, et al. (1998). "SAP90 binds and clusters kainate receptors causing incomplete desensitization". Neuron. 21 (4): 727–39....

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Phospholamban
Senin, 2025-10-27 23:06:46

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Calcium-induced calcium release
Minggu, 2025-12-14 19:42:50

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Buphenine
Minggu, 2025-12-21 15:18:41

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Annexin A5
Minggu, 2025-12-14 08:41:37

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Levomethorphan
Sabtu, 2026-05-16 03:12:24

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Sarcosine
Rabu, 2026-04-22 15:53:58

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Argiotoxin
Kamis, 2025-11-27 11:29:57

receptors: AMPA, NMDA (argiotoxin has higher potency at NMDA receptors), kainate, and nicotine acetylcholine receptors. It is thought that polyamine toxins'...

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Dexoxadrol
Sabtu, 2025-12-27 07:10:24

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Excitatory amino acid receptor agonist
Rabu, 2025-10-08 16:54:23

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Calretinin
Senin, 2026-05-11 10:45:45

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Isoflurane
Sabtu, 2026-05-09 08:41:45

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Plazinemdor
Sabtu, 2026-06-06 12:22:37

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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EVT-101
Selasa, 2025-12-23 14:38:03

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Methorphan
Selasa, 2026-03-31 21:35:26

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Calmodulin
Selasa, 2026-04-21 17:54:49

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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5,7-Dichlorokynurenic acid
Rabu, 2026-02-18 00:27:57

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Oxiracetam
Sabtu, 2026-06-06 15:50:04

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Dextrallorphan
Sabtu, 2025-12-27 07:24:45

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Methoxmetamine
Sabtu, 2025-12-27 07:18:40

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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ACE mixture
Senin, 2026-05-11 15:46:14

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Zonampanel
Selasa, 2025-12-23 14:00:31

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Methoxetamine
Rabu, 2026-05-20 13:28:18

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Troponin C
Jumat, 2026-06-05 16:41:16

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Dehydroepiandrosterone sulfate
Selasa, 2026-04-07 07:34:24

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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N-Ethylnorketamine
Sabtu, 2025-12-27 07:17:43

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Neramexane
Sabtu, 2025-12-27 07:09:34

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ryanodine receptor
Kamis, 2026-06-04 02:16:08

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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XW10508
Minggu, 2026-03-15 13:56:46

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Calpain
Sabtu, 2023-08-26 20:24:17

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Homoquinolinic acid
Kamis, 2026-05-14 06:36:57

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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N-Acetylaspartic acid
Selasa, 2026-03-10 18:09:40

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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LIN7B
Selasa, 2025-10-21 22:47:19

P, Choquet D, Lambert M, Mège RM, Mulle C (2002). "Recruitment of the kainate receptor subunit glutamate receptor 6 by cadherin/catenin complexes". J...

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Leteprinim
Sabtu, 2025-12-27 19:06:28

Middlemiss PJ, et al. (June 2001). "AIT-082 is neuroprotective against kainate-induced neuronal injury in rats". Experimental Neurology. 169 (2): 392–9...

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Arketamine
Rabu, 2026-05-06 05:01:45

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Calgranulin
Rabu, 2025-05-28 07:02:54

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Rhynchophylline
Selasa, 2025-04-29 11:53:50

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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PICK1
Rabu, 2025-07-16 05:09:40

Couthino V (February 2003). "Rapid and differential regulation of AMPA and kainate receptors at hippocampal mossy fibre synapses by PICK1 and GRIP". Neuron...

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CX-546
Senin, 2025-12-29 19:52:08

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Pentamidine
Minggu, 2025-10-05 03:41:26

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Racemorphan
Sabtu, 2025-12-27 07:25:32

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Mark Mayer
Selasa, 2025-02-18 13:42:47

permeability; analysis of the permeation and block of Ca permeable AMPA and kainate receptors by cytoplasmic polyamines; and structural studies on ligand binding...

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Levorphanol
Jumat, 2025-12-26 15:06:39

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Tetrazolylglycine
Selasa, 2025-12-23 14:30:22

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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GRIP1 (gene)
Kamis, 2025-07-17 23:46:27

Couthino V (February 2003). "Rapid and differential regulation of AMPA and kainate receptors at hippocampal mossy fibre synapses by PICK1 and GRIP". Neuron...

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Calreticulin
Rabu, 2026-05-27 20:37:15

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Noribogaine
Selasa, 2026-06-02 14:49:32

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Fibulin
Minggu, 2023-01-29 04:58:26

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Chloral hydrate/magnesium sulfate/pentobarbital
Sabtu, 2023-01-28 12:05:10

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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List of investigational antipsychotics
Jumat, 2026-06-05 11:45:16

LY-450108) – ionotropic glutamate AMPA receptor agonists, ionotropic glutamate kainate receptor antagonists, and metabotropic glutamate mGlu2 receptor modulators...

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Estradiol valerate/prasterone enanthate
Selasa, 2025-12-23 07:50:47

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Haloperidol decanoate
Rabu, 2026-01-14 05:01:39

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Glutamatergic
Selasa, 2026-05-05 02:59:28

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Perzinfotel
Jumat, 2026-04-03 11:32:14

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Reelin
Selasa, 2026-05-26 18:48:49

chain-migrating neuroblasts failed to detach properly. Moreover, in a kainate-induced mouse epilepsy model, exogenous reelin had prevented GCD, according...

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CGP-37849
Selasa, 2025-12-30 00:29:09

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Intracellular calcium-sensing proteins
Jumat, 2023-05-12 03:00:04

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Piretanide
Sabtu, 2026-04-11 10:28:46

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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PCPr
Senin, 2026-05-04 19:38:53

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Neboglamine
Selasa, 2025-12-23 12:53:34

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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TCTHP
Sabtu, 2025-12-27 09:00:36

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Fanapanel
Selasa, 2025-12-23 14:02:09

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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GRIA4
Senin, 2025-10-27 23:15:10

ionotropic AMPA glutamate receptor subunits (Glur2, Glur3, Glur4) and Kainate receptor subunits (Glur5, Glur6). Glutamate-gated ion channels are made...

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Caroverine
Selasa, 2025-12-23 14:03:02

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Nortilidine
Jumat, 2025-10-03 05:51:35

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Crocetin
Kamis, 2025-04-17 21:32:41

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Isoxsuprine
Minggu, 2025-12-21 15:18:22

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ketobemidone
Jumat, 2025-12-26 11:31:19

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Zelquistinel
Jumat, 2026-06-05 08:03:53

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Cyclopropane
Kamis, 2026-05-28 09:52:42

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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PEAQX
Senin, 2024-09-23 12:29:54

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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CX-516
Senin, 2025-12-29 19:51:56

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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ACPD
Senin, 2025-12-29 22:53:34

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Glufimet
Minggu, 2025-12-21 13:02:14

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Serine
Selasa, 2026-05-12 19:07:34

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Pomaglumetad
Kamis, 2026-06-04 09:13:48

other metabotropic glutamate receptors, ionotropic NMDA receptors, or kainate receptors, nor does it appear to have any affinity for adrenergic,...

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Long-term video-EEG monitoring
Jumat, 2026-01-16 04:52:26

A; Crutison, J; Thippeswamy, T (2015). "Immediate Epileptogenesis after Kainate-Induced Status Epilepticus in C57BL/6J Mice: Evidence from Long Term Continuous...

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3-MeO-PCE
Senin, 2026-05-04 19:38:41

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Quinolinic acid
Senin, 2026-02-02 21:29:36

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Deudextromethorphan/quinidine
Rabu, 2025-02-26 07:30:23

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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8A-PDHQ
Sabtu, 2025-12-27 07:11:39

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Methoxphenidine
Selasa, 2026-05-05 23:15:43

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Calnexin
Senin, 2025-05-19 09:03:18

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Aceglutamide
Sabtu, 2025-10-11 23:13:15

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Blarcamesine
Sabtu, 2026-05-30 12:39:13

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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3-MeO-PCP
Jumat, 2026-01-30 10:06:11

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Tabernanthine
Selasa, 2025-11-18 11:09:59

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Conantokin
Sabtu, 2025-12-06 16:58:04

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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CX614
Selasa, 2025-12-30 00:37:47

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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RAP-219
Minggu, 2026-05-31 14:36:31

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ephenidine
Sabtu, 2026-02-14 15:41:57

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Becampanel
Selasa, 2025-12-23 13:49:25

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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2-hydroxy-dATP diphosphatase
Minggu, 2025-11-23 05:55:31

oxidative damage of nucleic acids in the hippocampal microglia during kainate-induced excitotoxicity". The Journal of Neuroscience. 26 (6): 1688–98....

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Methoxyketamine
Sabtu, 2025-12-27 07:18:53

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Calexcitin
Senin, 2023-12-04 02:10:50

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Rapastinel
Kamis, 2026-06-04 09:02:34

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Eticyclidine
Senin, 2026-05-04 19:38:45

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Traxoprodil
Sabtu, 2026-02-28 12:08:10

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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2,2,2-Trichloroethanol
Rabu, 2025-08-20 08:50:58

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Glutamate transporter
Jumat, 2026-02-13 11:15:18

Norepinephrine transporters Serotonin transporters NMDA receptors AMPA receptors Kainate receptors Metabotropic glutamate receptors Ganel R, Rothstein JD (1999)...

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Ralfinamide
Senin, 2026-02-23 19:33:52

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Flufenamic acid
Jumat, 2026-01-30 05:29:00

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Etoxadrol
Jumat, 2026-05-15 12:59:28

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Felbamate
Kamis, 2026-05-21 03:08:37

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Arylcyclohexylamine
Sabtu, 2026-02-21 12:50:05

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Prasterone sulfate
Selasa, 2025-12-23 08:46:27

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Synaptotagmin
Rabu, 2025-11-26 23:30:12

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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ORG-26576
Selasa, 2025-12-23 11:54:52

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Tenocyclidine
Sabtu, 2025-12-27 07:23:01

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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CX717
Senin, 2026-01-26 13:55:07

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Osteonectin
Rabu, 2025-05-28 23:43:22

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Licostinel
Selasa, 2025-12-23 14:28:25

the NMDA receptor, licostinel also acts as an antagonist of the AMPA and kainate receptors at high concentrations (Kb = 0.9 μM and 2.5 μM, respectively)...

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Midafotel
Sabtu, 2025-12-27 07:09:55

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Synaptic pharmacology
Jumat, 2025-10-10 16:56:13

AM-251 GABAA bicuculline, gabazine GABAB CGP-54626 glycine strychnine kainate R .. metabotropic GluR, broad MCPG, pertussis toxin, NEM muscarinic AChR...

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MTEP
Rabu, 2025-12-31 18:30:19

effects of MTEP, a selective mGluR5 antagonists and neuropeptide Y on the kainate-induced toxicity in primary neuronal cultures". Pharmacological Reports...

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Metapramine
Rabu, 2025-12-24 12:24:01

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Selfotel
Senin, 2026-03-02 08:46:45

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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S-18986
Rabu, 2025-12-24 10:37:22

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Indantadol
Minggu, 2025-11-02 12:25:27

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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FBLN1
Kamis, 2025-07-17 23:33:54

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Methoxisopropamine
Sabtu, 2026-01-31 13:31:31

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ifenprodil
Senin, 2026-03-02 13:19:02

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Apical dendrite
Selasa, 2026-03-17 03:12:33

neurons have been found vulnerable to excitotoxic action of glutamate at the kainate receptor. These receptors are most dense in sectors CA3 and CA2 of the...

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Aptiganel
Sabtu, 2026-01-31 04:53:38

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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3-HO-PCP
Senin, 2026-05-04 19:38:39

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Patrizia Casaccia
Sabtu, 2026-04-18 05:08:48

methods of gene transfer in organotypic hippocampal brain slices to explore kainate receptor biology and electrophysiology. Her doctoral thesis explored sleep...

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S-Nitrosoglutathione
Rabu, 2025-12-31 22:43:17

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Post-transcriptional regulation
Minggu, 2026-05-24 06:03:30

GluR2, GluR3, GluR4, GluR5 and GluR6 (which are components of the AMPA and kainate receptors), the serotonin2C receptor, the GABA-alpha3 receptor subunit...

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Coronaridine
Minggu, 2026-05-17 02:06:11

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Kaitocephalin
Minggu, 2025-12-21 23:15:51

ionotropic. The ionotropic receptors are further divided into NMDA, AMPA, and kainate receptors. Kaitocephalin is a potent competitive antagonist of both NMDA...

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1,3-Diaminopropane
Senin, 2026-02-09 02:50:22

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Milnacipran
Rabu, 2026-06-03 03:07:56

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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2-Methyl-6-(phenylethynyl)pyridine
Senin, 2025-12-29 22:23:49

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Gavestinel
Senin, 2023-08-14 03:40:33

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Budipine
Selasa, 2026-06-02 14:48:31

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Milacemide
Rabu, 2025-11-26 07:35:29

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Apolipoprotein D
Sabtu, 2026-06-06 12:33:38

Rassart E (August 2017). "Apolipoprotein D Overexpression Protects Against Kainate-Induced Neurotoxicity in Mice". Molecular Neurobiology. 54 (6): 3948–3963...

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Hippocalcin
Jumat, 2026-02-20 06:16:20

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Irampanel
Selasa, 2025-12-23 14:23:52

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Levomethadone
Selasa, 2025-12-23 12:24:05

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Annexin A2
Selasa, 2025-10-21 05:01:44

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Glutathione disulfide
Minggu, 2025-11-23 05:30:27

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Gacyclidine
Sabtu, 2025-12-27 07:23:06

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Cystine/glutamate transporter
Kamis, 2025-10-02 15:36:04

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Besonprodil
Kamis, 2024-09-05 03:54:30

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Prasterone enanthate
Selasa, 2025-12-23 08:37:53

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Esmethadone
Selasa, 2025-12-23 12:23:47

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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PD-137889
Sabtu, 2025-12-27 08:57:28

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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PEPA (drug)
Sabtu, 2026-01-10 22:01:15

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Gelsolin
Kamis, 2026-03-26 16:33:54

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Remacemide
Minggu, 2026-04-19 18:21:38

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Levomilnacipran
Rabu, 2026-06-03 03:01:08

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Ibogamine
Jumat, 2025-12-26 20:09:14

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Rislenemdaz
Jumat, 2026-03-13 06:58:53

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Regucalcin
Rabu, 2025-10-22 09:42:10

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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MAP3K10
Jumat, 2025-07-18 00:20:40

PMID 11076863. Savinainen A, Garcia EP, Dorow D, Marshall J, Liu YF (2001). "Kainate receptor activation induces mixed lineage kinase-mediated cellular signaling...

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Sabeluzole
Kamis, 2026-01-01 03:06:39

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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4-MeO-PCP
Jumat, 2026-01-30 10:06:17

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Sodium- and chloride-dependent glycine transporter 1
Sabtu, 2026-02-14 14:03:20

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Dieticyclidine
Sabtu, 2025-12-27 07:21:54

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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IDRA-21
Rabu, 2025-12-24 10:18:04

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Gerald Fischbach
Jumat, 2026-04-10 21:30:53

injections to apply glutamate and other agonists including NMDA, AMPA, and kainate to different regions of the neurons, he noticed that certain hot spots...

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Α-Endopsychosin
Kamis, 2025-08-28 16:33:50

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Excitatory amino acid receptor antagonist
Rabu, 2025-10-08 16:51:36

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Hodgkinsine
Senin, 2025-12-29 20:46:13

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Cyclic ADP-ribose
Selasa, 2025-09-30 11:04:17

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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AMN082
Jumat, 2025-12-26 22:29:21

are fast-acting ligand-gated ion channels and include AMPA receptors, kainate receptors, and NMDA receptors. Metabotropic receptors are G-protein coupled...

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Hypericin
Kamis, 2026-06-04 16:51:40

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Calcium-binding protein
Sabtu, 2024-01-27 06:56:58

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Neuronal calcium sensor
Jumat, 2026-02-20 06:13:23

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Dalzanemdor
Jumat, 2026-06-05 07:48:26

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Clinical neurochemistry
Selasa, 2026-05-05 02:57:00

receptors of neurotransmitters include AMPA receptors, NMDA receptors, and Kainate Receptors. Changes in the homeostatic levels of many neurologically active...

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Nicotinic acid adenine dinucleotide phosphate
Senin, 2025-10-13 09:58:57

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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2-MDP
Sabtu, 2025-12-27 07:11:45

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Dexanabinol
Senin, 2025-11-17 01:29:34

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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4-Chlorokynurenine
Selasa, 2025-12-23 12:01:56

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Alaproclate
Jumat, 2026-04-03 10:39:30

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Rolicyclidine
Senin, 2026-05-04 19:38:58

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Norketamine
Sabtu, 2025-12-27 07:19:10

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Nitromemantine
Jumat, 2026-01-30 10:31:01

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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LY-503430
Rabu, 2025-12-24 10:37:11

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Omigapil
Kamis, 2026-01-29 05:16:38

withdrawal, and lactacystin. Additionally, omigapil can prevent NMDA and kainate receptor excitotoxicity in rat cortical neurons as well as toxicity from...

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Fluorolintane
Sabtu, 2025-12-27 07:34:37

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Homocysteic acid
Kamis, 2026-02-05 02:20:32

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Prasterone
Rabu, 2026-01-28 07:20:45

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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AP-7 (drug)
Jumat, 2025-12-26 22:29:37

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Oncomodulin
Rabu, 2025-01-01 13:43:21

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Testosterone propionate/testosterone cypionate/prasterone
Sabtu, 2023-03-11 07:32:12

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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7-Chlorokynurenic acid
Rabu, 2026-02-18 00:21:35

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Alazocine
Jumat, 2026-01-02 10:56:02

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Pregnenolone succinate
Selasa, 2025-12-23 10:10:16

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Fourphit
Sabtu, 2025-12-27 08:45:55

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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LY-235959
Rabu, 2025-12-31 02:17:40

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Parkin (protein)
Minggu, 2025-10-05 06:58:46

SCF-like ubiquitin ligase complex and protects postmitotic neurons from kainate excitotoxicity". Neuron. 37 (5): 735–49. doi:10.1016/s0896-6273(03)00084-9...

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Sarcalumenin
Selasa, 2026-03-24 06:07:47

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Pesampator
Selasa, 2025-12-23 11:54:48

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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S100G
Rabu, 2025-10-22 11:58:33

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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3-MeO-PCMo
Senin, 2026-05-04 19:38:43

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Talampanel
Minggu, 2026-03-01 08:39:41

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Tulrampator
Selasa, 2025-12-23 11:54:27

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Hydroxynorketamine
Minggu, 2026-03-15 13:56:35

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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N-Acetylaspartylglutamic acid
Minggu, 2025-12-28 22:39:51

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Metaphit
Sabtu, 2025-12-27 08:45:47

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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LY-404187
Rabu, 2025-12-24 10:38:59

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Niflumic acid
Senin, 2025-12-01 13:05:00

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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Recoverin
Minggu, 2025-10-05 00:04:45

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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FBLN2
Kamis, 2025-02-20 15:10:23

Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...

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Lubeluzole
Senin, 2025-12-29 21:05:13

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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L-687,384
Jumat, 2025-12-26 11:47:17

Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...

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