Search Results: Kainate
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Kainate receptor
Rabu, 2025-12-24 11:13:18Kainate receptors, or kainic acid receptors (KARs), are ionotropic receptors that respond to the neurotransmitter glutamate. They were first identified...
Click to read more »Kainic acid
Rabu, 2026-04-22 10:42:31Kainic acid, or kainate, is an acid that naturally occurs in some seaweed. Kainic acid is a potent neuroexcitatory amino acid agonist that acts by activating...
Click to read more »5-Fluorowillardiine
Kamis, 2026-05-28 06:07:33selective agonist for the AMPA receptor, with only limited effects at the kainate receptor. It is an excitotoxic neurotoxin when used in vivo and so is rarely...
Click to read more »GRIK5
Rabu, 2025-10-22 02:32:04Glutamate receptor, ionotropic kainate 5 is a protein that in humans is encoded by the GRIK5 gene. This gene encodes a protein that belongs to the glutamate-gated...
Click to read more »Glutamate (neurotransmitter)
Minggu, 2026-05-24 14:36:01receptors, and metabotropic glutamate receptors. A fourth class, known as kainate receptors, are similar in many respects to AMPA receptors, but much less...
Click to read more »GYKI 52466
Rabu, 2025-12-24 11:46:49receptor antagonist (IC50 values are 10-20, ~ 450 and >> 50 μM for AMPA-, kainate- and NMDA-induced responses respectively), orally-active anticonvulsant...
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Selasa, 2026-02-24 06:02:47Glutamate ionotropic receptor kainate type subunit 2, also known as ionotropic glutamate receptor 6 or GluR6, is a protein that in humans is encoded by...
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Sabtu, 2026-04-04 03:50:57receptors: AMPA and kainate receptors. Willardiine analogs have been developed that have different binding affinities for the AMPA and kainate receptors. These...
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Rabu, 2025-12-24 09:39:37of the AMPA and kainate subtypes of the ionotropic glutamate receptor family, with selectivity for the GluR5 subtype of the kainate receptor. It has...
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Sabtu, 2025-07-19 02:21:07selective agonist for the kainate receptor. This potent agonist has nearly 3,000 fold- and 200-fold selectivity for kainate receptors over AMPA and NMDA...
Click to read more »Ionotropic glutamate receptor
Sabtu, 2026-04-11 21:51:59binding properties (pharmacology) and sequence similarity: AMPA receptors, kainate receptors, NMDA receptors and delta receptors (see below). AMPA receptors...
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Senin, 2026-01-05 14:04:50Glutamate receptor, ionotropic, kainate 1, also known as GRIK1, is a protein that in humans is encoded by the GRIK1 gene. This gene encodes one of the...
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Kamis, 2025-10-16 01:36:37isolate the action of other glutamate receptors in the brain, i.e., AMPA and kainate receptors. AP5 can block the conversion of a silent synapse to an active...
Click to read more »5-Iodowillardiine
Sabtu, 2026-05-30 18:49:47a selective agonist for some kainate receptor subunits with only limited effects at AMPA receptors. It activates kainate receptors containing GluK1 (GluR5)...
Click to read more »Riluzole
Selasa, 2026-05-26 06:39:37damaged neurons. Riluzole has also been reported to directly inhibit the kainate and NMDA receptors. The drug has also been shown to postsynaptically potentiate...
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Selasa, 2025-12-23 14:03:47AMPA receptors in micromolar concentrations (~10–20 μM) and also blocks kainate receptors. In experiments, it is used to counter glutamate excitotoxicity...
Click to read more »N-Methyl-D-aspartic acid
Kamis, 2025-12-11 05:00:07has no effect on other glutamate receptors (such as those for AMPA and kainate). NMDA receptors are particularly important when they become overactive...
Click to read more »Quisqualic acid
Jumat, 2026-02-06 12:55:00Quisqualic acid is an agonist of the AMPA, kainate, and group I metabotropic glutamate receptors. It is one of the most potent AMPA receptor agonists...
Click to read more »NS102
Kamis, 2024-09-26 21:07:26NS102 is a kainate receptor antagonist. NS102 at Sigma-Aldrich Johansen, Tina H; Drejer, Joergen; Watjen, Frank; Nielsen, Elsebet O (1993). "A novel non-NMDA...
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Rabu, 2026-05-20 13:40:50and II metabotropic glutamate receptors, and weakly activating AMPA and kainate receptors. Taken systemically, it is a prodrug of muscimol, broken down...
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Senin, 2026-04-13 19:24:27especially potent at kainate receptors and AMPA receptors, with inhibitory potencies summarised in the table: The inhibition of kainate receptors by NPTX-8...
Click to read more »GRIK4
Kamis, 2025-07-17 00:27:42GRIK4 (glutamate receptor, ionotropic, kainate 4) is a kainate receptor subtype belonging to the family of ligand-gated ion channels which is encoded...
Click to read more »CNQX
Selasa, 2025-12-23 14:04:19cyanquixaline (6-cyano-7-nitroquinoxaline-2,3-dione) is a competitive AMPA/kainate receptor antagonist. Its chemical formula is C9H4N4O4. CNQX is often used...
Click to read more »Juan Lerma Gómez
Selasa, 2026-03-10 08:48:18its role in health and disease. He described the existence of functional kainate receptors (KARs) in central neurons and applied single-cell RT-PCR to study...
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Sabtu, 2026-03-28 19:09:21and 5-HT3 receptors, and as a negative allosteric modulator of the AMPA, kainate, and NMDA receptors, as well as of nicotinic acetylcholine receptors. Clinically...
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Rabu, 2026-05-27 21:56:16Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Kamis, 2026-01-29 23:47:46types of ionotropic glutamate receptors, the other two being AMPA and kainate receptors. Depending on its subunit composition, its ligands are glutamate...
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Selasa, 2025-12-23 14:28:44pharmacologically active, acting as a negative allosteric modulator of the AMPA and kainate receptors and as an inhibitor of vesicular glutamate transporters. It also...
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Sabtu, 2026-05-23 21:27:32ionotropic glutamate receptors in the micromolar range, including the AMPA and kainate receptors and, to a lesser extent, the NMDA receptor. It acts as an antagonist...
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Selasa, 2026-04-07 07:34:24lesser extent, it also acts as a negative allosteric modulator of the AMPA, kainate, and glycine receptors, and may interact with the nACh receptors as well...
Click to read more »Neuron
Sabtu, 2026-05-30 00:03:48is a G-protein coupled receptor (often referred to as GPCR). AMPA and Kainate receptors function as cation channels permeable to Na+ cation channels...
Click to read more »Dextromethorphan
Kamis, 2026-04-02 19:40:24et al. (April 2005). "The dextromethorphan analog dimemorfan attenuates kainate-induced seizures via sigma1 receptor activation: comparison with the effects...
Click to read more »Glutamate receptor
Rabu, 2026-05-20 22:20:23plasticity. They are activated by the drug kainate and are permeable to both sodium and potassium ions. Kainate receptors are expressed in a variety of brain...
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Sabtu, 2025-12-27 09:00:03Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Kynurenic acid
Rabu, 2026-03-04 00:39:59to act on five targets: As an antagonist at ionotropic AMPA, NMDA and Kainate glutamate receptors in the concentration range of 0.1-2.5 mM. As a noncompetitive...
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Sabtu, 2025-12-27 08:32:51Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Sabtu, 2026-05-02 23:36:24post-synaptic neuron will be increased. Direct blockade of glutamatergic AMPA and kainate receptors are also believed to contribute to the hypnotic/anticonvulsant...
Click to read more »Diazoxide
Minggu, 2026-05-31 11:04:06hyperinsulinism. Diazoxide acts as a positive allosteric modulator of the AMPA and kainate receptors, suggesting potential application as a cognitive enhancer. Diazoxide...
Click to read more »Reversal potential
Sabtu, 2025-12-20 20:44:18neurotransmitter receptors including glutamate receptors (AMPA, NMDA, and kainate), nicotinic acetylcholine (nACh), and serotonin (5-HT3) receptors are nonselective...
Click to read more »Β-Methylamino-L-alanine
Senin, 2026-03-09 11:24:09excitotoxin on glutamate receptors, such as NMDA, calcium-dependent AMPA, and kainate receptors. The activation of the metabotropic glutamate receptor 5 is believed...
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Kamis, 2026-05-07 03:55:27weak agonist of the glycine receptor and of both NMDA and non-NMDA (AMPA/kainate) ionotropic glutamate receptors. It has been proposed to be a potential...
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Selasa, 2025-07-15 11:13:27Glutamate receptor, ionotropic kainate 3 is a protein that in humans is encoded by the GRIK3 gene. This gene encodes a protein that belongs to the ligand-gated...
Click to read more »Quisqualamine
Minggu, 2025-12-21 17:15:08vitro. The NMDA receptor antagonists magnesium and DL-AP5, the AMPA and kainate receptor antagonist CNQX, and the GABAB receptor antagonist 2-hydroxysaclofen...
Click to read more »Barbiturate
Selasa, 2026-04-28 05:16:03In addition to this GABAergic effect, barbiturates also block AMPA and kainate receptors, subtypes of ionotropic glutamate receptor. Glutamate is the...
Click to read more »Furosemide
Jumat, 2026-05-22 17:55:16Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Hexobarbital
Jumat, 2025-03-21 22:45:52inhibitory effect, hexobarbital blocks, like all barbiturates, AMPA receptors, kainate receptors, neural acetylcholine receptors. And above all, barbiturates...
Click to read more »AMPA receptor
Rabu, 2026-05-06 12:02:46"Structure of a glutamate-receptor ligand-binding core in complex with kainate". Nature. 395 (6705): 913–7. Bibcode:1998Natur.395..913A. doi:10.1038/27692...
Click to read more »F-17475
Sabtu, 2026-02-21 12:50:13Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Phenidone
Minggu, 2026-05-03 23:26:53Myung-Bok; Kim, Won-Ki; Ko, Kwang Ho (August 18, 2000). "Phenidone prevents kainate-induced neurotoxicity via antioxidant mechanisms". Brain Research. 874...
Click to read more »Atomoxetine
Selasa, 2026-06-02 14:48:14Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Glutamine
Sabtu, 2026-01-10 19:31:32Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »UBP-302
Jumat, 2026-01-02 00:04:02UBP-302 is a highly selective kainate receptor antagonist used in the study of many neurological processes. It is active at micromolar concentration within...
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Jumat, 2026-06-05 15:37:48neurons increase with intense visual stimuli. Animal models suggest that kainate signaling negatively regulates serotonin actions in the retina, with possible...
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Kamis, 2026-05-07 21:34:49blocks NMDAR and β2-subunit-containing nACh channels, weakly inhibits AMPA, kainate, GABAC and 5-HT3 receptors, and slightly potentiates GABAA and glycine...
Click to read more »Glossary of neuroscience
Rabu, 2026-01-21 21:24:09processing during sleep. Kainate receptor A subtype of ionotropic glutamate receptor involved in fast excitatory synaptic transmission. Kainate receptors play roles...
Click to read more »List of investigational headache and migraine drugs
Jumat, 2026-06-05 11:36:24– migraine [77] Dasolampanel (NGX-426) – ionotropic glutamate AMPA and kainate receptor antagonist – migraine [78] Dextromethorphan/quinidine (DXM/Q;...
Click to read more »Trifluoromethyldeschloroketamine
Sabtu, 2025-12-27 09:01:33Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Methadone
Selasa, 2026-06-02 22:13:18Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Senin, 2026-05-04 19:38:35Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Selasa, 2026-02-17 23:56:19Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Senin, 2026-02-23 11:15:53Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Minggu, 2026-06-07 05:07:29Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Senin, 2026-04-13 03:17:56Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Kamis, 2026-02-12 03:56:47Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »SGK1
Selasa, 2026-02-24 06:07:42role of SGK1 in memory consolidation. "SGK isoforms upregulate AMPA and kainate receptors and thus are expected to enhance the excitatory effects of glutamate"...
Click to read more »Diphenidine
Sabtu, 2026-02-14 15:30:54Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Kamis, 2026-04-02 22:11:23Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Rabu, 2026-01-07 06:44:28Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Rabu, 2026-05-27 04:14:54receptor signaling in the ventral tegmental area are mediated by AMPA/kainate receptors". American Journal of Physiology. Endocrinology and Metabolism...
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Minggu, 2026-05-17 22:18:27Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Rabu, 2026-02-25 02:52:02Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »G protein-coupled receptor
Senin, 2026-06-01 17:51:25receptor, 5-HT3 serotonin receptor and glutamate receptors (NMDAR, AMPAR and kainate receptor), which are ion channels. Regulation of immune system activity...
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Jumat, 2026-01-30 21:53:59Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Dextropropoxyphene
Selasa, 2026-06-02 14:48:46Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Kamis, 2026-03-26 02:34:58Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Rabu, 2026-04-22 10:43:25and amygdaloid nucleus. It damages the neurons by activating AMPA and kainate receptors, causing an influx of calcium. Although calcium flowing into...
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Sabtu, 2025-05-24 05:36:54Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Halothane
Selasa, 2026-01-27 04:51:36activates 5-HT3 and twin-pore K+ channels. It does not affect the AMPA or kainate receptors. Halothane (2-bromo-2-chloro-1,1,1-trifluoroethane) is a very...
Click to read more »Methylene blue
Jumat, 2026-05-22 06:54:00Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Rabu, 2026-06-03 16:35:07Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »List of investigational tinnitus drugs
Kamis, 2026-05-14 06:57:15[13] Selurampanel (BGG-492; BGG-492A) – ionotropic glutamate AMPA and kainate receptor antagonist [14] Sodium phenylbutyrate slow-release (4-PB-D-alanin;...
Click to read more »Lacosamide
Selasa, 2026-05-19 21:16:52abnormal neuronal connections in the brain. Lacosamide does not affect AMPA, kainate, NMDA, GABAA, GABAB or a variety of dopaminergic, serotonergic, adrenergic...
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Kamis, 2026-05-28 23:46:44acids Glutamate Glu, E Metabotropic glutamate receptors NMDA receptors, kainate receptors, AMPARs Small: Amino acids Gamma-aminobutyric acid GABA GABAB...
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Sabtu, 2026-05-23 07:49:18Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Jumat, 2026-05-08 01:06:57Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Selasa, 2025-10-14 23:26:55during seizure — Evidence from 13C-enrichment of extracellular glutamate in kainate rat model". PLOS ONE. 12 (4) e0174845. Bibcode:2017PLoSO..1274845K. doi:10...
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Kamis, 2026-05-07 13:18:50GABAA, GABAB1a, GABAB1δ, GABAB2, GABAA-rho Glutamatergic: NMDA, AMPA, Kainate, mGluR1, mGluR2, mGluR3, mGluR4, mGluR5, mGluR6, mGluR7 Glycinergic: Glycine...
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Rabu, 2026-05-06 00:38:18Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Minggu, 2026-02-08 03:05:21Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Minggu, 2026-03-15 13:51:43Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Rabu, 2026-05-27 04:46:05channels, high-voltage-activated calcium channels, GABAA receptors, AMPA/kainate receptors, and carbonic anhydrase isoenzymes. There is evidence that topiramate...
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Sabtu, 2026-02-14 03:50:17blocks NMDAR and β2-subunit-containing nACh channels, weakly inhibits AMPA, kainate, GABAC and 5-HT3 receptors, and slightly potentiates GABAA and glycine...
Click to read more »Teresa Puthussery
Minggu, 2026-04-26 08:34:20Venkataramani, S., Gayet-Primo, J., Grünert, U., & Taylor, W. R. (2014). Kainate Receptors Mediate Synaptic Input to Transient and Sustained OFF Visual...
Click to read more »BQ-869
Rabu, 2026-04-22 14:42:05Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Senin, 2026-03-16 00:30:08Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Sabtu, 2025-07-19 12:48:06Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
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Minggu, 2026-05-31 10:59:29electroshock, electrical kindling of the amygdala, pentylenetetrazol, kainate, NMDA, and picrotoxin. Researchers hoped this wide-ranging activity would...
Click to read more »3-Fluorodeschloroketamine
Sabtu, 2025-12-27 08:21:51Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Selasa, 2026-05-19 10:08:25(α-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid), NMDA (N-methyl-D-aspartate) and kainate subtypes of ionotropic glutamate receptors follows. It is the activation...
Click to read more »Hydrochlorothiazide
Rabu, 2026-05-13 18:25:57Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Senin, 2026-05-11 06:30:11Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Selasa, 2026-06-02 15:32:44Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Rabu, 2025-12-24 09:55:44that cyclothiazide is a positive allosteric modulator of the AMPA and kainate receptors, capable of reducing or essentially eliminating rapid desensitization...
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Senin, 2026-02-09 11:46:37Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Sabtu, 2026-02-21 12:27:28Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Kamis, 2025-12-18 19:07:59positive regulation of excitatory postsynaptic potential regulation of kainate selective glutamate receptor activity Sources:Amigo / QuickGO Orthologs...
Click to read more »Selurampanel
Jumat, 2026-01-30 10:03:52quinoxalinedione series which acts as a competitive antagonist of the AMPA and kainate receptors and, as of 2015, is being investigated in clinical trials by...
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Minggu, 2026-03-22 15:00:46Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Gunnar Svaetichin
Rabu, 2025-10-01 04:51:33(March 1984). "Hyperpolarization of fish retinal horizontal cells by kainate and quisqualate". Nature. 308 (5957): 360–362. Bibcode:1984Natur.308..360H...
Click to read more »Acromelic acid A
Kamis, 2025-07-17 22:08:38Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Senin, 2026-05-04 19:38:33Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Kamis, 2026-05-28 07:16:07Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Fluorexetamine
Sabtu, 2025-12-27 08:20:30Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Xenon
Selasa, 2026-06-02 01:14:34Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Calcium signaling
Kamis, 2026-06-04 02:04:03Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Acetylcysteine
Kamis, 2026-04-02 02:17:58Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Radu Aricescu
Rabu, 2025-10-01 12:01:01complexes", Science, vol. 353, issue 6296 (2016). "Transsynaptic Modulation of Kainate Receptor Functions by C1q-like Proteins", Neuron, vol. 90, issue 4 (2016)...
Click to read more »Meprobamate
Rabu, 2026-02-04 14:24:32Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Carisoprodol
Selasa, 2026-05-05 06:04:28Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »3-Methyl-PCP
Sabtu, 2025-12-27 08:31:39Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Zinc
Jumat, 2026-06-05 21:56:22Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Syntenin-1
Jumat, 2025-07-18 01:31:12Couthino V (February 2003). "Rapid and differential regulation of AMPA and kainate receptors at hippocampal mossy fibre synapses by PICK1 and GRIP". Neuron...
Click to read more »Neurocalcin
Jumat, 2026-02-20 06:15:35Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Piracetam
Kamis, 2026-03-26 03:39:30Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Hemantane
Sabtu, 2026-03-14 19:21:08Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Allopregnanolone
Selasa, 2026-05-12 05:45:06no action at other ligand-gated ion channels, including the NMDA, AMPA, kainate, and glycine receptors. Unlike progesterone, allopregnanolone is inactive...
Click to read more »Xanthurenic acid
Selasa, 2025-12-23 12:02:44Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Dimemorfan
Kamis, 2025-05-29 21:18:05et al. (April 2005). "The dextromethorphan analog dimemorfan attenuates kainate-induced seizures via sigma1 receptor activation: comparison with the effects...
Click to read more »2-Bromodeschloroketamine
Sabtu, 2025-12-27 08:34:01Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Esketamine
Sabtu, 2026-05-02 02:22:03Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Convulsant
Rabu, 2026-02-04 13:01:58in animals as it is a cyclic analog of l-glutamate and an agonist for kainate receptors in the brain which makes it a potent neurotoxin and excitant...
Click to read more »NEFA (drug)
Sabtu, 2025-12-27 07:09:49Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Haloperidol
Selasa, 2026-06-02 14:49:07Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Dizocilpine
Senin, 2026-04-27 11:28:08Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Alexei Verkhratsky
Senin, 2026-03-02 11:40:51Kettenmann, H.; Verkhratsky, A. (1997). "Na+/Ca2+ exchanger modulates kainate-triggered Ca2+ signaling in Bergmann glial cells in situ". FASEB J. 11...
Click to read more »Amnesic shellfish poisoning
Sabtu, 2024-09-14 16:11:48and amygdaloid nucleus. It damages the neurons by activating AMPA and kainate receptors, causing an influx of calcium. Although calcium flowing into...
Click to read more »Magnesium
Kamis, 2026-05-28 20:39:07Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Eliprodil
Senin, 2026-05-11 13:59:45Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »DLG4
Kamis, 2025-07-31 20:47:58Couthino V (February 2003). "Rapid and differential regulation of AMPA and kainate receptors at hippocampal mossy fibre synapses by PICK1 and GRIP". Neuron...
Click to read more »EVT-103
Jumat, 2024-01-05 14:19:53Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Deoxymethoxetamine
Sabtu, 2025-12-27 08:35:25Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »GRIA2
Senin, 2025-10-27 23:17:06specifically the ionotropic AMPA receptor subunits (GluR2, GluR3, GluR4) and kainate receptor subunits (GluR5, GluR6). Glutamate-gated ion channels are composed...
Click to read more »Nitric oxide
Selasa, 2026-05-26 13:14:18Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Biological neuron model
Selasa, 2026-05-12 12:06:45kinetic currents. Four neurotransmitters primarily influence the CNS. AMPA/kainate receptors are fast excitatory mediators while NMDA receptors mediate considerably...
Click to read more »Annexin
Kamis, 2026-01-01 08:54:05Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Dextromethorphan/bupropion
Kamis, 2026-06-04 15:43:12Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Alcohol (drug)
Senin, 2026-06-01 02:31:31Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Glycine
Senin, 2026-04-27 18:18:56Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Dimethylglycine
Senin, 2026-05-04 00:02:11Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Alanine
Kamis, 2026-04-30 13:17:28Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Phencyclidine
Jumat, 2026-05-15 14:16:34Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Philanthotoxin
Jumat, 2026-01-30 09:58:45Philanthotoxins reversibly inhibit AMPA (also called the "quisqualate receptor"), kainate, and NMDA ionotropic glutamate receptors (iGluRs). Philanthotoxins have...
Click to read more »Blixeprodil
Senin, 2026-05-04 19:48:10Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Toluene
Jumat, 2026-04-24 10:24:19Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Dasolampanel
Selasa, 2025-12-23 14:23:19analog of tezampanel and thereby competitive antagonist of the AMPA and kainate receptors which was under development by Raptor Pharmaceuticals/Torrey...
Click to read more »Putrescine
Senin, 2026-01-26 14:51:19Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Edward Boyden
Selasa, 2026-05-19 06:02:11high-efficacy soma-targeted opsin through combining the N-terminal 150 residues of kainate receptor subunit 2 (KA2) to the high-photocurrent channelrhodopsin CoChR...
Click to read more »L-701324
Sabtu, 2025-12-27 19:02:22Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Theanne Griffith
Sabtu, 2025-12-27 01:11:16Swanson G (2015). "Identification of critical functional determinants of kainate receptor modulation by auxiliary protein Neto2". Journal of Physiology...
Click to read more »Tramadol
Jumat, 2026-05-29 05:45:43Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Farampator
Kamis, 2026-06-04 09:25:58Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »S-phase kinase-associated protein 1
Sabtu, 2025-07-19 14:21:56SCF-like ubiquitin ligase complex and protects postmitotic neurons from kainate excitotoxicity". Neuron. 37 (5): 735–49. doi:10.1016/s0896-6273(03)00084-9...
Click to read more »3-Methyl-PCPy
Sabtu, 2025-12-27 08:51:12Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »GRID2
Minggu, 2025-12-28 20:07:35glutamate receptors. They possess 14–24% sequence homology with AMPA, kainate, and NMDA subunits, but, despite their name, have been found not to directly...
Click to read more »CX1739
Senin, 2026-03-30 14:10:56Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Chromosome 21
Minggu, 2025-09-28 04:19:32protein 3A, mitochondrial GRIK1: encoding glutamate receptor ionotropic, kainate 1 H2BC12L: encoding histone H2B type F-S HLCS: encoding enzyme holocarboxylase...
Click to read more »Northern blot
Jumat, 2026-01-02 02:42:24Zukin, R. S. (1993). "Developmental Regulation of mRNAs Encoding Rat Brain Kainate/AMPA Receptors: A Northern Analysis Study". J. Neurochem. 61 (6): 2239–2246...
Click to read more »L-687,414
Sabtu, 2026-02-21 15:01:44Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Long-term depression
Sabtu, 2026-05-30 04:20:50α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid receptors (AMPARs), kainate receptors (KARs), and metabotropic glutamate receptors (mGluRs) during...
Click to read more »Mibampator
Selasa, 2025-12-23 11:54:57Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Diethylenetriamine
Jumat, 2026-06-05 14:21:21Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Inhalational anesthetic
Rabu, 2026-05-13 06:02:09Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »AMPA receptor positive allosteric modulator
Selasa, 2025-12-23 11:54:16Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Pentobarbital
Rabu, 2026-05-20 22:50:26Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »DNQX
Selasa, 2025-12-23 14:04:077-dinitroquinoxaline-2,3-dione) is a competitive antagonist at AMPA and kainate receptors, two ionotropic glutamate receptor (iGluR) subfamilies. It is...
Click to read more »Channel blocker
Rabu, 2025-12-24 13:02:13Channel blockers are also known to act at AMPA receptors, Glycine receptors, Kainate receptors, P2X receptors and Zinc (Zn2+)-activated channels. The type of...
Click to read more »ACEA-1328
Rabu, 2025-12-24 23:52:43Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Hydroxetamine
Sabtu, 2025-12-27 08:47:28Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »1-Aminocyclopropane-1-carboxylic acid
Senin, 2025-11-24 05:28:30Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Pharmacology of ethanol
Minggu, 2026-04-05 14:07:08negative allosteric modulator AMPA receptor: negative allosteric modulator Kainate receptor: negative allosteric modulator Glycine receptor: positive allosteric...
Click to read more »Lanicemine
Rabu, 2025-12-24 11:08:21Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »3-Chloro-PCP
Minggu, 2026-05-17 02:28:14Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Kynurenine
Kamis, 2026-03-12 04:56:20Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Farah Lubin
Minggu, 2026-04-12 18:59:26expression and transcriptional regulation in the hippocampus. She found that kainate, a glutamate analog, elicited activation of NF-κB via the classical IkB...
Click to read more »Spermine
Sabtu, 2026-02-21 22:41:33Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Ketamine/temsirolimus
Jumat, 2025-02-28 12:11:07Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »AMPA
Selasa, 2025-02-11 02:25:59Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Trichloroethylene
Kamis, 2026-06-04 09:43:04Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Deschloroketamine
Sabtu, 2025-12-27 08:34:36Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Radiprodil
Senin, 2026-01-26 14:02:36Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Minocycline
Kamis, 2026-06-04 16:40:01Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »NYX-2925
Senin, 2026-02-23 11:52:45Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Excitatory synapse
Kamis, 2025-09-18 06:51:07postsynaptic receptors including the NMDA receptor, AMPA receptor, and kainate receptors. These receptors are all cation channels that allow positively...
Click to read more »3-Fluoro-PCP
Senin, 2026-05-04 19:38:37Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Bumetanide
Selasa, 2026-03-03 01:57:01Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »GRIA3
Senin, 2025-10-27 23:16:02ionotropic AMPA glutamate receptor subunits (GluA2, GluA3, GluA4) and kainate receptor subunits (GluK1, GluK2). Glutamate gated ion channels are made...
Click to read more »Receptor (biochemistry)
Sabtu, 2026-05-16 00:35:41Receptors G protein Exogenous Ligand Glutamate iGluRs: NMDA, AMPA, and Kainate receptors Na+, K+, Ca2+ Ketamine Glutamate receptors: mGluRs Gq or Gi/o...
Click to read more »Cytidine
Selasa, 2026-04-07 12:17:09Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Silent synapse
Senin, 2026-03-30 07:56:17(AMPARs) (formerly known as quisqualate receptors), NMDA receptors (NMDARs), kainate receptors, and metabotropic glutamate receptors (mGluRs). Most research...
Click to read more »S100 protein
Sabtu, 2025-10-04 15:18:15Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »NPDPA
Sabtu, 2026-02-21 18:47:24Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Orphenadrine
Selasa, 2026-06-02 14:49:37Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Excitatory amino acid receptor ligand
Jumat, 2024-03-22 12:39:12Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »HA-966
Minggu, 2025-12-21 15:58:19Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Nooglutyl
Kamis, 2026-06-04 01:03:58Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Cyclic glycine-proline
Minggu, 2025-12-21 13:13:58Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Methoxyflurane
Sabtu, 2026-02-21 17:05:10Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Methoxpropamine
Kamis, 2026-01-01 17:31:19Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Annexin A1
Senin, 2025-11-17 11:25:01Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »18-Methoxycoronaridine
Senin, 2026-05-11 19:16:26Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »1,1,1-Trichloroethane
Jumat, 2026-02-27 20:03:58Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Oligodendrocyte progenitor cell
Sabtu, 2025-10-04 23:28:52proteoglycan-positive oligodendrocyte precursor cells in the normal and kainate-lesioned rat hippocampus". Neuroscience. 92 (1): 83–95. doi:10.1016/S0306-4522(98)00751-9...
Click to read more »Ketofol
Rabu, 2025-05-28 23:27:11Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »2-FXPr
Sabtu, 2025-12-27 08:26:31Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Huperzine A
Minggu, 2026-05-17 02:28:01Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Halogenated ether
Jumat, 2026-05-15 22:56:07Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »FBXW7
Kamis, 2025-07-17 23:34:08SCF-like ubiquitin ligase complex and protects postmitotic neurons from kainate excitotoxicity". Neuron. 37 (5): 735–49. doi:10.1016/s0896-6273(03)00084-9...
Click to read more »Ligand-gated ion channel
Senin, 2025-10-27 23:27:58HBGR2 GLUA3, GluR3, GluRC, GluR-C, GluR-K3 GLUA4, GluR4, GluRD, GluR-D Kainate GluK GluK1 GluK2 GluK3 GluK4 GluK5 GRIK1 GRIK2 GRIK3 GRIK4 GRIK5 GLUK5...
Click to read more »List of investigational substance-related disorder drugs
Jumat, 2026-06-05 08:37:19Tezampanel (LY-293558; NGX-424; PRN-001-01) – ionotropic glutamate AMPA and kainate receptor antagonist – opioid-related disorders TMP-301 (Heptares 25; HTL-0014242;...
Click to read more »Apigenin
Kamis, 2026-06-04 14:44:26Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Biology of bipolar disorder
Senin, 2026-05-25 04:45:44and neuronal morphology. The rACC demonstrates reduced expression NMDA, kainate and GABA related proteins. These findings may be compensating for increased...
Click to read more »Pramiracetam
Jumat, 2025-11-21 09:38:48Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Psychotridine
Rabu, 2025-12-24 12:05:45Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Membrane estrogen receptor
Kamis, 2026-05-21 15:53:46(February 1998). "Novel mechanism for non-genomic action of 17β-oestradiol on kainate-induced currents in isolated rat CA1 hippocampal neurones". The Journal...
Click to read more »Quinoxalinedione
Selasa, 2025-12-23 14:02:36for the diol tautomer. Quinoxalinediones act as antagonists of the AMPA, kainate, and/or NMDA receptors of the ionotropic glutamate receptor family. Examples...
Click to read more »Calbindin
Selasa, 2025-12-30 20:39:40Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »David Lodge (scientist)
Sabtu, 2024-10-19 19:40:04characterised its actions between AMPA, N-Methyl-D-aspartic acid (NMDA) and kainate receptor subtypes. At the Royal Veterinary College, Lodge linked his interests...
Click to read more »Agmatine
Senin, 2026-03-23 06:45:50Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Dextrorphan
Minggu, 2026-04-26 20:47:44Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Tyrosine phosphorylation
Sabtu, 2025-06-14 12:30:34receptors. These receptors can be divided into three major classes, AMPA, kainate, and NMDA receptors, based on their selective agonists and on their physiological...
Click to read more »Inositol trisphosphate
Senin, 2025-10-13 09:58:47Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Molecular neuroscience
Selasa, 2024-04-02 02:05:51concentrations. Ionotropic glutamate receptors can include NMDA, AMPA, and kainate receptors. These receptors are named after agonists that facilitate glutamate...
Click to read more »Lomerizine
Jumat, 2026-01-23 16:41:24protection against NMDA-induced and kainate-induced neurotoxicity. Lomerizine was shown to have little affinity for NMDA or kainate receptors, so its protectivity...
Click to read more »Bita Moghaddam
Rabu, 2026-05-13 23:32:16local activation of ionotropic glutamate receptors (AMPA receptors and kainate receptors). A few years later, she found that metabotropic glutamate receptors...
Click to read more »Changjoon Justin Lee
Selasa, 2025-12-23 09:01:11Reese Hospital, Columbia University Thesis The Expression and Function of Kainate and AMPA Receptors in Nociceptive Dorsal Root Ganglion Neurons (2001)...
Click to read more »Clavulanic acid
Sabtu, 2026-05-30 18:29:58Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Indeloxazine
Rabu, 2026-05-27 04:23:00Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »1,2-Diphenylethylamine
Sabtu, 2026-02-21 12:57:20Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Aniracetam
Minggu, 2025-03-30 22:17:03Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »ZD-9379
Senin, 2025-12-29 22:03:09Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Apimostinel
Senin, 2025-06-30 21:43:30Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »CGP-39551
Sabtu, 2025-12-27 02:50:18Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Ana Cristina Rego
Sabtu, 2026-06-06 02:02:43(11-12), 1405-1417 AC Rego, MW Ward, DG Nicholls. Mitochondria control ampa/kainate receptor-induced cytoplasmic calcium deregulation in rat cerebellar granule...
Click to read more »Dextromethorphan/quinidine
Senin, 2025-12-15 15:00:15Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Gliotransmitter
Senin, 2025-09-08 21:12:03cytosolic Ca2+ concentrations in astrocytes. Its main target receptors include Kainate receptors, metabotropic glutamate receptors (mGluRs), and especially N-methyl...
Click to read more »Microglia
Rabu, 2026-05-20 14:41:29Christensen RN, Ha BK, Sun F, Bresnahan JC, Beattie MS (July 2006). "Kainate induces rapid redistribution of the actin cytoskeleton in ameboid microglia"...
Click to read more »Osteocalcin
Rabu, 2026-04-22 21:36:11Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Cycloserine
Rabu, 2026-05-27 15:25:19Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Stephen Heinemann
Jumat, 2025-07-18 01:28:11Heinemann contributed to differentiating: AMPA receptors, NMDA receptors, and kainate receptors. As shown by Heinemann, NMDA receptors differ in that they allow...
Click to read more »Perampanel
Kamis, 2026-05-14 14:50:07Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »PCPEP
Sabtu, 2025-12-27 08:56:13Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Ampakine
Rabu, 2025-12-24 08:38:37Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Pre-Bötzinger complex
Selasa, 2026-04-07 06:23:58studies showed that excitatory transmission, predominantly via AMPA- and kainate-type ionotropic glutamate receptors were essential for rhythm generation...
Click to read more »Delucemine
Sabtu, 2025-12-27 07:10:55Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »GRIA1
Senin, 2025-10-27 23:16:292003). "Heteromer formation of delta2 glutamate receptors with AMPA or kainate receptors". Brain Res. Mol. Brain Res. 110 (1): 27–37. doi:10.1016/s0169-328x(02)00561-2...
Click to read more »4-Keto-PCP
Sabtu, 2025-12-27 08:32:11Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »DLG3
Kamis, 2025-07-17 23:21:41Garcia EP, Mehta S, Blair LA, et al. (1998). "SAP90 binds and clusters kainate receptors causing incomplete desensitization". Neuron. 21 (4): 727–39....
Click to read more »Phospholamban
Senin, 2025-10-27 23:06:46Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Calcium-induced calcium release
Minggu, 2025-12-14 19:42:50Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Buphenine
Minggu, 2025-12-21 15:18:41Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Annexin A5
Minggu, 2025-12-14 08:41:37Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Levomethorphan
Sabtu, 2026-05-16 03:12:24Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Sarcosine
Rabu, 2026-04-22 15:53:58Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Argiotoxin
Kamis, 2025-11-27 11:29:57receptors: AMPA, NMDA (argiotoxin has higher potency at NMDA receptors), kainate, and nicotine acetylcholine receptors. It is thought that polyamine toxins'...
Click to read more »Dexoxadrol
Sabtu, 2025-12-27 07:10:24Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Excitatory amino acid receptor agonist
Rabu, 2025-10-08 16:54:23Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Calretinin
Senin, 2026-05-11 10:45:45Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Isoflurane
Sabtu, 2026-05-09 08:41:45Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Plazinemdor
Sabtu, 2026-06-06 12:22:37Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »EVT-101
Selasa, 2025-12-23 14:38:03Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Methorphan
Selasa, 2026-03-31 21:35:26Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Calmodulin
Selasa, 2026-04-21 17:54:49Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »5,7-Dichlorokynurenic acid
Rabu, 2026-02-18 00:27:57Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Oxiracetam
Sabtu, 2026-06-06 15:50:04Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Dextrallorphan
Sabtu, 2025-12-27 07:24:45Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Methoxmetamine
Sabtu, 2025-12-27 07:18:40Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »ACE mixture
Senin, 2026-05-11 15:46:14Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Zonampanel
Selasa, 2025-12-23 14:00:31Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Methoxetamine
Rabu, 2026-05-20 13:28:18Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Troponin C
Jumat, 2026-06-05 16:41:16Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Dehydroepiandrosterone sulfate
Selasa, 2026-04-07 07:34:24Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »N-Ethylnorketamine
Sabtu, 2025-12-27 07:17:43Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Neramexane
Sabtu, 2025-12-27 07:09:34Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Ryanodine receptor
Kamis, 2026-06-04 02:16:08Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »XW10508
Minggu, 2026-03-15 13:56:46Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Calpain
Sabtu, 2023-08-26 20:24:17Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Homoquinolinic acid
Kamis, 2026-05-14 06:36:57Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »N-Acetylaspartic acid
Selasa, 2026-03-10 18:09:40Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »LIN7B
Selasa, 2025-10-21 22:47:19P, Choquet D, Lambert M, Mège RM, Mulle C (2002). "Recruitment of the kainate receptor subunit glutamate receptor 6 by cadherin/catenin complexes". J...
Click to read more »Leteprinim
Sabtu, 2025-12-27 19:06:28Middlemiss PJ, et al. (June 2001). "AIT-082 is neuroprotective against kainate-induced neuronal injury in rats". Experimental Neurology. 169 (2): 392–9...
Click to read more »Arketamine
Rabu, 2026-05-06 05:01:45Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Calgranulin
Rabu, 2025-05-28 07:02:54Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Rhynchophylline
Selasa, 2025-04-29 11:53:50Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »PICK1
Rabu, 2025-07-16 05:09:40Couthino V (February 2003). "Rapid and differential regulation of AMPA and kainate receptors at hippocampal mossy fibre synapses by PICK1 and GRIP". Neuron...
Click to read more »CX-546
Senin, 2025-12-29 19:52:08Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Pentamidine
Minggu, 2025-10-05 03:41:26Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Racemorphan
Sabtu, 2025-12-27 07:25:32Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Mark Mayer
Selasa, 2025-02-18 13:42:47permeability; analysis of the permeation and block of Ca permeable AMPA and kainate receptors by cytoplasmic polyamines; and structural studies on ligand binding...
Click to read more »Levorphanol
Jumat, 2025-12-26 15:06:39Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Tetrazolylglycine
Selasa, 2025-12-23 14:30:22Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »GRIP1 (gene)
Kamis, 2025-07-17 23:46:27Couthino V (February 2003). "Rapid and differential regulation of AMPA and kainate receptors at hippocampal mossy fibre synapses by PICK1 and GRIP". Neuron...
Click to read more »Calreticulin
Rabu, 2026-05-27 20:37:15Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Noribogaine
Selasa, 2026-06-02 14:49:32Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Fibulin
Minggu, 2023-01-29 04:58:26Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Chloral hydrate/magnesium sulfate/pentobarbital
Sabtu, 2023-01-28 12:05:10Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »List of investigational antipsychotics
Jumat, 2026-06-05 11:45:16LY-450108) – ionotropic glutamate AMPA receptor agonists, ionotropic glutamate kainate receptor antagonists, and metabotropic glutamate mGlu2 receptor modulators...
Click to read more »Estradiol valerate/prasterone enanthate
Selasa, 2025-12-23 07:50:47Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Haloperidol decanoate
Rabu, 2026-01-14 05:01:39Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Glutamatergic
Selasa, 2026-05-05 02:59:28Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Perzinfotel
Jumat, 2026-04-03 11:32:14Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Reelin
Selasa, 2026-05-26 18:48:49chain-migrating neuroblasts failed to detach properly. Moreover, in a kainate-induced mouse epilepsy model, exogenous reelin had prevented GCD, according...
Click to read more »CGP-37849
Selasa, 2025-12-30 00:29:09Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Intracellular calcium-sensing proteins
Jumat, 2023-05-12 03:00:04Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Piretanide
Sabtu, 2026-04-11 10:28:46Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »PCPr
Senin, 2026-05-04 19:38:53Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Neboglamine
Selasa, 2025-12-23 12:53:34Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »TCTHP
Sabtu, 2025-12-27 09:00:36Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Fanapanel
Selasa, 2025-12-23 14:02:09Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »GRIA4
Senin, 2025-10-27 23:15:10ionotropic AMPA glutamate receptor subunits (Glur2, Glur3, Glur4) and Kainate receptor subunits (Glur5, Glur6). Glutamate-gated ion channels are made...
Click to read more »Caroverine
Selasa, 2025-12-23 14:03:02Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Nortilidine
Jumat, 2025-10-03 05:51:35Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Crocetin
Kamis, 2025-04-17 21:32:41Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Isoxsuprine
Minggu, 2025-12-21 15:18:22Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Ketobemidone
Jumat, 2025-12-26 11:31:19Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Zelquistinel
Jumat, 2026-06-05 08:03:53Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Cyclopropane
Kamis, 2026-05-28 09:52:42Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »PEAQX
Senin, 2024-09-23 12:29:54Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »CX-516
Senin, 2025-12-29 19:51:56Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »ACPD
Senin, 2025-12-29 22:53:34Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Glufimet
Minggu, 2025-12-21 13:02:14Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Serine
Selasa, 2026-05-12 19:07:34Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Pomaglumetad
Kamis, 2026-06-04 09:13:48other metabotropic glutamate receptors, ionotropic NMDA receptors, or kainate receptors, nor does it appear to have any affinity for adrenergic,...
Click to read more »Long-term video-EEG monitoring
Jumat, 2026-01-16 04:52:26A; Crutison, J; Thippeswamy, T (2015). "Immediate Epileptogenesis after Kainate-Induced Status Epilepticus in C57BL/6J Mice: Evidence from Long Term Continuous...
Click to read more »3-MeO-PCE
Senin, 2026-05-04 19:38:41Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Quinolinic acid
Senin, 2026-02-02 21:29:36Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Deudextromethorphan/quinidine
Rabu, 2025-02-26 07:30:23Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »8A-PDHQ
Sabtu, 2025-12-27 07:11:39Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Methoxphenidine
Selasa, 2026-05-05 23:15:43Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Calnexin
Senin, 2025-05-19 09:03:18Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Aceglutamide
Sabtu, 2025-10-11 23:13:15Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Blarcamesine
Sabtu, 2026-05-30 12:39:13Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »3-MeO-PCP
Jumat, 2026-01-30 10:06:11Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Tabernanthine
Selasa, 2025-11-18 11:09:59Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Conantokin
Sabtu, 2025-12-06 16:58:04Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »CX614
Selasa, 2025-12-30 00:37:47Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »RAP-219
Minggu, 2026-05-31 14:36:31Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Ephenidine
Sabtu, 2026-02-14 15:41:57Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Becampanel
Selasa, 2025-12-23 13:49:25Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »2-hydroxy-dATP diphosphatase
Minggu, 2025-11-23 05:55:31oxidative damage of nucleic acids in the hippocampal microglia during kainate-induced excitotoxicity". The Journal of Neuroscience. 26 (6): 1688–98....
Click to read more »Methoxyketamine
Sabtu, 2025-12-27 07:18:53Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Calexcitin
Senin, 2023-12-04 02:10:50Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Rapastinel
Kamis, 2026-06-04 09:02:34Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Eticyclidine
Senin, 2026-05-04 19:38:45Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Traxoprodil
Sabtu, 2026-02-28 12:08:10Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »2,2,2-Trichloroethanol
Rabu, 2025-08-20 08:50:58Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Glutamate transporter
Jumat, 2026-02-13 11:15:18Norepinephrine transporters Serotonin transporters NMDA receptors AMPA receptors Kainate receptors Metabotropic glutamate receptors Ganel R, Rothstein JD (1999)...
Click to read more »Ralfinamide
Senin, 2026-02-23 19:33:52Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Flufenamic acid
Jumat, 2026-01-30 05:29:00Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Etoxadrol
Jumat, 2026-05-15 12:59:28Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Felbamate
Kamis, 2026-05-21 03:08:37Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Arylcyclohexylamine
Sabtu, 2026-02-21 12:50:05Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Prasterone sulfate
Selasa, 2025-12-23 08:46:27Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Synaptotagmin
Rabu, 2025-11-26 23:30:12Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »ORG-26576
Selasa, 2025-12-23 11:54:52Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Tenocyclidine
Sabtu, 2025-12-27 07:23:01Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »CX717
Senin, 2026-01-26 13:55:07Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Osteonectin
Rabu, 2025-05-28 23:43:22Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Licostinel
Selasa, 2025-12-23 14:28:25the NMDA receptor, licostinel also acts as an antagonist of the AMPA and kainate receptors at high concentrations (Kb = 0.9 μM and 2.5 μM, respectively)...
Click to read more »Midafotel
Sabtu, 2025-12-27 07:09:55Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Synaptic pharmacology
Jumat, 2025-10-10 16:56:13AM-251 GABAA bicuculline, gabazine GABAB CGP-54626 glycine strychnine kainate R .. metabotropic GluR, broad MCPG, pertussis toxin, NEM muscarinic AChR...
Click to read more »MTEP
Rabu, 2025-12-31 18:30:19effects of MTEP, a selective mGluR5 antagonists and neuropeptide Y on the kainate-induced toxicity in primary neuronal cultures". Pharmacological Reports...
Click to read more »Metapramine
Rabu, 2025-12-24 12:24:01Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Selfotel
Senin, 2026-03-02 08:46:45Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »S-18986
Rabu, 2025-12-24 10:37:22Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Indantadol
Minggu, 2025-11-02 12:25:27Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »FBLN1
Kamis, 2025-07-17 23:33:54Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Methoxisopropamine
Sabtu, 2026-01-31 13:31:31Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Ifenprodil
Senin, 2026-03-02 13:19:02Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Apical dendrite
Selasa, 2026-03-17 03:12:33neurons have been found vulnerable to excitotoxic action of glutamate at the kainate receptor. These receptors are most dense in sectors CA3 and CA2 of the...
Click to read more »Aptiganel
Sabtu, 2026-01-31 04:53:38Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »3-HO-PCP
Senin, 2026-05-04 19:38:39Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Patrizia Casaccia
Sabtu, 2026-04-18 05:08:48methods of gene transfer in organotypic hippocampal brain slices to explore kainate receptor biology and electrophysiology. Her doctoral thesis explored sleep...
Click to read more »S-Nitrosoglutathione
Rabu, 2025-12-31 22:43:17Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Post-transcriptional regulation
Minggu, 2026-05-24 06:03:30GluR2, GluR3, GluR4, GluR5 and GluR6 (which are components of the AMPA and kainate receptors), the serotonin2C receptor, the GABA-alpha3 receptor subunit...
Click to read more »Coronaridine
Minggu, 2026-05-17 02:06:11Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Kaitocephalin
Minggu, 2025-12-21 23:15:51ionotropic. The ionotropic receptors are further divided into NMDA, AMPA, and kainate receptors. Kaitocephalin is a potent competitive antagonist of both NMDA...
Click to read more »1,3-Diaminopropane
Senin, 2026-02-09 02:50:22Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Milnacipran
Rabu, 2026-06-03 03:07:56Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »2-Methyl-6-(phenylethynyl)pyridine
Senin, 2025-12-29 22:23:49Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Gavestinel
Senin, 2023-08-14 03:40:33Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Budipine
Selasa, 2026-06-02 14:48:31Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Milacemide
Rabu, 2025-11-26 07:35:29Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Apolipoprotein D
Sabtu, 2026-06-06 12:33:38Rassart E (August 2017). "Apolipoprotein D Overexpression Protects Against Kainate-Induced Neurotoxicity in Mice". Molecular Neurobiology. 54 (6): 3948–3963...
Click to read more »Hippocalcin
Jumat, 2026-02-20 06:16:20Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Irampanel
Selasa, 2025-12-23 14:23:52Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Levomethadone
Selasa, 2025-12-23 12:24:05Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Annexin A2
Selasa, 2025-10-21 05:01:44Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Glutathione disulfide
Minggu, 2025-11-23 05:30:27Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Gacyclidine
Sabtu, 2025-12-27 07:23:06Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Cystine/glutamate transporter
Kamis, 2025-10-02 15:36:04Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Besonprodil
Kamis, 2024-09-05 03:54:30Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Prasterone enanthate
Selasa, 2025-12-23 08:37:53Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Esmethadone
Selasa, 2025-12-23 12:23:47Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »PD-137889
Sabtu, 2025-12-27 08:57:28Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »PEPA (drug)
Sabtu, 2026-01-10 22:01:15Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Gelsolin
Kamis, 2026-03-26 16:33:54Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Remacemide
Minggu, 2026-04-19 18:21:38Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Levomilnacipran
Rabu, 2026-06-03 03:01:08Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Ibogamine
Jumat, 2025-12-26 20:09:14Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Rislenemdaz
Jumat, 2026-03-13 06:58:53Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Regucalcin
Rabu, 2025-10-22 09:42:10Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »MAP3K10
Jumat, 2025-07-18 00:20:40PMID 11076863. Savinainen A, Garcia EP, Dorow D, Marshall J, Liu YF (2001). "Kainate receptor activation induces mixed lineage kinase-mediated cellular signaling...
Click to read more »Sabeluzole
Kamis, 2026-01-01 03:06:39Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »4-MeO-PCP
Jumat, 2026-01-30 10:06:17Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Sodium- and chloride-dependent glycine transporter 1
Sabtu, 2026-02-14 14:03:20Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Dieticyclidine
Sabtu, 2025-12-27 07:21:54Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »IDRA-21
Rabu, 2025-12-24 10:18:04Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Gerald Fischbach
Jumat, 2026-04-10 21:30:53injections to apply glutamate and other agonists including NMDA, AMPA, and kainate to different regions of the neurons, he noticed that certain hot spots...
Click to read more »Α-Endopsychosin
Kamis, 2025-08-28 16:33:50Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Excitatory amino acid receptor antagonist
Rabu, 2025-10-08 16:51:36Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Hodgkinsine
Senin, 2025-12-29 20:46:13Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Cyclic ADP-ribose
Selasa, 2025-09-30 11:04:17Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »AMN082
Jumat, 2025-12-26 22:29:21are fast-acting ligand-gated ion channels and include AMPA receptors, kainate receptors, and NMDA receptors. Metabotropic receptors are G-protein coupled...
Click to read more »Hypericin
Kamis, 2026-06-04 16:51:40Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Calcium-binding protein
Sabtu, 2024-01-27 06:56:58Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Neuronal calcium sensor
Jumat, 2026-02-20 06:13:23Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Dalzanemdor
Jumat, 2026-06-05 07:48:26Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Clinical neurochemistry
Selasa, 2026-05-05 02:57:00receptors of neurotransmitters include AMPA receptors, NMDA receptors, and Kainate Receptors. Changes in the homeostatic levels of many neurologically active...
Click to read more »Nicotinic acid adenine dinucleotide phosphate
Senin, 2025-10-13 09:58:57Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »2-MDP
Sabtu, 2025-12-27 07:11:45Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Dexanabinol
Senin, 2025-11-17 01:29:34Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »4-Chlorokynurenine
Selasa, 2025-12-23 12:01:56Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Alaproclate
Jumat, 2026-04-03 10:39:30Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Rolicyclidine
Senin, 2026-05-04 19:38:58Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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Sabtu, 2025-12-27 07:19:10Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Nitromemantine
Jumat, 2026-01-30 10:31:01Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »LY-503430
Rabu, 2025-12-24 10:37:11Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Omigapil
Kamis, 2026-01-29 05:16:38withdrawal, and lactacystin. Additionally, omigapil can prevent NMDA and kainate receptor excitotoxicity in rat cortical neurons as well as toxicity from...
Click to read more »Fluorolintane
Sabtu, 2025-12-27 07:34:37Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Homocysteic acid
Kamis, 2026-02-05 02:20:32Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Prasterone
Rabu, 2026-01-28 07:20:45Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »AP-7 (drug)
Jumat, 2025-12-26 22:29:37Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Oncomodulin
Rabu, 2025-01-01 13:43:21Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Testosterone propionate/testosterone cypionate/prasterone
Sabtu, 2023-03-11 07:32:12Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »7-Chlorokynurenic acid
Rabu, 2026-02-18 00:21:35Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Alazocine
Jumat, 2026-01-02 10:56:02Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Pregnenolone succinate
Selasa, 2025-12-23 10:10:16Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Fourphit
Sabtu, 2025-12-27 08:45:55Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »LY-235959
Rabu, 2025-12-31 02:17:40Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Parkin (protein)
Minggu, 2025-10-05 06:58:46SCF-like ubiquitin ligase complex and protects postmitotic neurons from kainate excitotoxicity". Neuron. 37 (5): 735–49. doi:10.1016/s0896-6273(03)00084-9...
Click to read more »Sarcalumenin
Selasa, 2026-03-24 06:07:47Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Pesampator
Selasa, 2025-12-23 11:54:48Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »S100G
Rabu, 2025-10-22 11:58:33Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »3-MeO-PCMo
Senin, 2026-05-04 19:38:43Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Talampanel
Minggu, 2026-03-01 08:39:41Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Tulrampator
Selasa, 2025-12-23 11:54:27Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Hydroxynorketamine
Minggu, 2026-03-15 13:56:35Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »N-Acetylaspartylglutamic acid
Minggu, 2025-12-28 22:39:51Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Metaphit
Sabtu, 2025-12-27 08:45:47Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »LY-404187
Rabu, 2025-12-24 10:38:59Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Niflumic acid
Senin, 2025-12-01 13:05:00Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »Recoverin
Minggu, 2025-10-05 00:04:45Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »FBLN2
Kamis, 2025-02-20 15:10:23Ligand-gated 5-HT3 receptor Ionotropic glutamate receptors AMPA receptors Kainate receptors NMDA receptors P2X receptors Voltage-gated L N P R T TRP channels...
Click to read more »Lubeluzole
Senin, 2025-12-29 21:05:13Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
Click to read more »L-687,384
Jumat, 2025-12-26 11:47:17Sevoflurane Talampanel; Unknown/unsorted antagonists: Minocycline KARTooltip Kainate receptor Agonists: Main site agonists: 5-Bromowillardiine 5-Iodowillardiine...
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